SCHEMBL8352120

SCHEMBL8352120

CCOC(=O)c1ncn(C)c1C(=O)OCC

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
APOBEC3A P31941 1/20 0.50
APOBEC3G Q9HC16 1/20 0.50
ALDH1A1 P00352 5/20 0.47
MAPT P10636 2/20 0.47
GABRA1 P14867 7/20 0.45
GABRG2 P18507 7/20 0.45
GABRB3 P28472 7/20 0.45
GABRA5 P31644 7/20 0.45
GABRA3 P34903 7/20 0.45
GABRA2 P47869 7/20 0.45
KMT2A Q03164 2/20 0.44
HPGD P15428 3/20 0.43
KDM4E B2RXH2 2/20 0.43
HSD17B10 Q99714 2/20 0.43
GABRA6 Q16445 5/20 0.43
GABRB2 P47870 3/20 0.43
HTT P42858 1/20 0.42
GABRA4 P48169 2/20 0.42
CYP1A2 P05177 2/20 0.42
CYP2D6 P10635 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5937208 0.84 ALDH1A1 (0.47) APOBEC3AAPOBEC3GALDH1A1MAPTKMT2A
SCHEMBL5727138 0.84 ALDH1A1 (0.48) APOBEC3AAPOBEC3GALDH1A1MAPTGABRA1
SCHEMBL14710629 0.81 KMT2A (0.42) APOBEC3AAPOBEC3GALDH1A1MAPTKMT2A
SCHEMBL22697032 0.81 MAPK1 (0.43) APOBEC3AAPOBEC3GALDH1A1MAPTKMT2A
SCHEMBL4355684 0.81 LMNA (0.46) APOBEC3AAPOBEC3GALDH1A1MAPTKMT2A
SCHEMBL23769132 0.81 ALDH1A1 (0.46) APOBEC3AAPOBEC3GALDH1A1MAPTGABRA1
SCHEMBL1990691 0.81 ALDH1A1 (0.46) APOBEC3AAPOBEC3GALDH1A1MAPTGABRA1
SCHEMBL31553574 0.81 ALDH1A1 (0.49) ALDH1A1MAPTHPGDKDM4EHSD17B10
SCHEMBL11656354 0.80 ALDH1A1 (0.48) ALDH1A1MAPTGABRA1GABRA5HPGD
SCHEMBL29173554 0.79 ALDH1A1 (0.44) APOBEC3AAPOBEC3GALDH1A1MAPTGABRA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 22 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12370192-B2 Azole-fused pyridazin-3(2H)-one derivatives TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2025-07-29 US disclosed
US-20250066369-A1 BICYCLIC PHTHALAZIN-1(2H)-ONE DERIVATIVES AND RELATED USES NodThera Limited (GB) 2025-02-27 US disclosed
EP-4460505-A1 BICYCLIC PHTHALAZIN-1(2H)-ONE DERIVATIVES AND RELATED USES Nodthera Limited (GB) 2024-11-13 EP disclosed
CN-118922421-A Bicyclic phthalazin-1 (2H) -one derivatives and related uses 诺瑟拉有限公司 2024-11-08 CN disclosed
EP-4031552-B1 AZOLE-FUSED PYRIDAZIN-3(2H)-ONE DERIVATIVES TAKEDA PHARMACEUTICALS CO (JP) 2024-11-06 EP disclosed
WO-2023133271-A1 BICYCLIC PHTHALAZIN-1(2H)-ONE DERIVATIVES AND RELATED USES NodThera Limited (GB) 2023-07-13 WO disclosed
US-20230028114-A1 AZOLE-FUSED PYRIDAZIN-3(2H)-ONE DERIVATIVES TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2023-01-26 US disclosed
US-20230028114-A1 AZOLE-FUSED PYRIDAZIN-3(2H)-ONE DERIVATIVES TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2023-01-26 US disclosed
EP-4031552-A1 AZOLE-FUSED PYRIDAZIN-3(2H)-ONE DERIVATIVES Takeda Pharmaceutical Company Limited (JP) 2022-07-27 EP disclosed
CN-114728975-A Azole-fused pyridazin-3 (2H) -one derivatives 武田药品工业株式会社 2022-07-08 CN disclosed
US-8367282-B2 Compound or its tautomer, metal complex compound, colored photosensitive curing composition, color filter, and production FUJIFILM CORPORATION (JP) 2013-02-05 US disclosed
US-8367282-B2 Compound or its tautomer, metal complex compound, colored photosensitive curing composition, color filter, and production FUJIFILM CORPORATION (JP) 2013-02-05 US disclosed
US-20120238752-A1 COMPOUND OR ITS TAUTOMER, METAL COMPLEX COMPOUND, COLORED PHOTOSENSITIVE CURING COMPOSITION, COLOR FILTER, AND PRODUCTION FUJIFILM CORPORATION (JP) 2012-09-20 US disclosed
US-8197994-B2 Colorant of a dipyrromethene-based metal complex obtained from a metal of iron, zinc, cobalt, copper or vanadium oxide and a dipyrromethene-based compound and a phthalocyanine dye FUJIFILM CORPORATION (JP) 2012-06-12 US disclosed
US-20120138877-A1 COMPOUND OR ITS TAUTOMER, METAL COMPLEX COMPOUND, COLORED PHOTOSENSITIVE CURING COMPOSITION, COLOR FILTER, AND PRODUCTION FUJIFILM CORPORATION (JP) 2012-06-07 US disclosed
US-20100230647-A1 COMPOUND OR ITS TAUTOMER, METAL COMPLEX COMPOUND, COLORED PHOTOSENSITIVE CURING COMPOSITION, COLOR FILTER, AND PRODUCTION FUJIFILM CORPORATION (JP) 2010-09-16 US disclosed
US-20080076044-A1 Compound or its tautomer, metal complex compound, colored photosensitive curing composition, color filter, and production FUJIFILM CORPORATION (JP) 2008-03-27 US disclosed
US-6004966-A ANTIISCHEMIC AGENTS; PYRAZOLO(3,4-D)PYRIMIDINDE, PURINE, ANDPTERIDINE DERIVATIVES BTG INTERNATIONAL LIMITED (GB) 1999-12-21 US disclosed
EP-0796099-A1 USE OF XANTHINE OXIDASE INHIBITORS AS ANTI-ISCHAEMIC AGENTS BTG INTERNATIONAL LIMITED (GB) 1997-09-24 EP disclosed
WO-1996017610-A1 USE OF XANTHINE OXIDASE INHIBITORS AS ANTI-ISCHAEMIC AGENTS BRITISH TECHNOLOGY GROUP LIMITED (GB) 1996-06-13 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230028114-A1 AZOLE-FUSED PYRIDAZIN-3(2H)-ONE DERIVATIVES GPR139, GPR119, GPR39 APOBEC3A 4848/4885APOBEC3G 4737/4885ALDH1A1 1955/4885
US-20250066369-A1 BICYCLIC PHTHALAZIN-1(2H)-ONE DERIVATIVES AND RELATED USES IL1B, NLRP3, IL1A APOBEC3A 4137/4885APOBEC3G 4313/4885ALDH1A1 401/4885
US-20120238752-A1 COMPOUND OR ITS TAUTOMER, METAL COMPLEX COMPOUND, COLORED PHOTOSENSITIVE CURING COMPOSITION, COLOR FILTER, AND PRODUCTION PBRM1, CRY1, MAPT APOBEC3A 2435/4885APOBEC3G 3142/4885ALDH1A1 1098/4885
US-12370192-B2 Azole-fused pyridazin-3(2H)-one derivatives GPR139, GPR119, GPR39 APOBEC3A 4848/4885APOBEC3G 4737/4885ALDH1A1 1955/4885
US-20100230647-A1 COMPOUND OR ITS TAUTOMER, METAL COMPLEX COMPOUND, COLORED PHOTOSENSITIVE CURING COMPOSITION, COLOR FILTER, AND PRODUCTION CRY1, IK, PRMT5 APOBEC3A 2311/4885APOBEC3G 3002/4885ALDH1A1 2769/4885
US-20080076044-A1 Compound or its tautomer, metal complex compound, colored photosensitive curing composition, color filter, and production PBRM1, CRY1, MAPT APOBEC3A 2435/4885APOBEC3G 3142/4885ALDH1A1 1098/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.