SCHEMBL8410035

SCHEMBL8410035

O=S(=O)([O-])c1cc(Nc2nc(Nc3ccccc3)nc(Nc3ccccc3)n2)ccc1/C=C/c1ccc(Nc2nc(Nc3ccccc3)nc(Nc3ccccc3)n2)cc1.[Na+]

nearest known ligand 0.55

Known targets — ChEMBL curated mechanism

ABCC8ACEADORA1ADORA2AADORA2BADORA3ALDH5A1ALOX5ALOX5APATP4AATP4BBRAFCA1CA12CA2CA4CYSLTR1DHFRDPEP1EDNRAEDNRBESR2F10FDPSFGF1GABBR1GABBR2GABRA1GABRA2GABRA3GABRA4GABRA5GABRA6GABRB1GABRB2GABRB3GABRDGABREGABRG1GABRG2GABRG3GABRPGABRQGARTGNRHRGSC1HMGCRIMPDH1IMPDH2KCNJ11LY96NOD2NR3C1NS3NS4ANS5bP2RY1P2RY12P2RY2P2RY4P2RY6PBP2XPDE3APDE3BPDE4APDE4BPDE4CPDE4DPDK1PDK2PDK3PDK4PPARGPPATPTGIRPTGS1PTGS2RAF1RYR1RYR3SCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASERPINC1SLC12A1SLC12A3SYKTHRATHRBTLR3TLR4TLR9TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYMSVKORC1XDHblablaIMP-1blaOXA-33blaOXA-58blaT-3blaT-4blaT-5blaT-6dacAdacBdacCfolAfolPfolP1ftsIfusAgaggyrAgyrBmecAmrcAmrcBmrdApbp1apbp1bpbp2pbp2apbp2bpbp3pbp4pbpApbpBpbpCpbpFpolponBrplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpoArpoBrpoCrpoZrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of None. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 known ✓ O43570 9/20 0.44
CA1 known ✓ P00915 9/20 0.44
CA2 known ✓ P00918 9/20 0.44
P2RY4 known ✓ P51582 2/20 0.40
THRB known ✓ P10828 1/20 0.40
P2RY12 known ✓ Q9H244 2/20 0.39
P2RY1 known ✓ P47900 1/20 0.39
P2RY2 known ✓ P41231 1/20 0.39
P2RY6 known ✓ Q15077 1/20 0.39
RAD51 Q06609 5/20 0.55
CA9 Q16790 9/20 0.44
APEX1 P27695 2/20 0.42
MEN1 O00255 1/20 0.40
USP2 O75604 1/20 0.40
LMNA P02545 1/20 0.40
TP53 P04637 1/20 0.40
POLB P06746 1/20 0.40
CYP3A4 P08684 1/20 0.40
GAA P10253 1/20 0.40
CYP2D6 P10635 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4821301 1.00 RAD51 (0.55) RAD51CA12CA1CA2CA9
SCHEMBL8410050 1.00 RAD51 (0.55) RAD51CA12CA1CA2CA9
SCHEMBL4821260 1.00 RAD51 (0.55) RAD51CA12CA1CA2CA9
SCHEMBL893765 0.95 RAD51 (0.60) RAD51CA12CA1CA2CA9
SCHEMBL29737199 0.95 RAD51 (0.60) RAD51CA12CA1CA2CA9
SCHEMBL1169584 0.95 RAD51 (0.60) RAD51CA12CA1CA2CA9
SCHEMBL30532269 0.95 RAD51 (0.60) RAD51CA12CA1CA2CA9
SCHEMBL4435900 0.89 RAD51 (0.54) RAD51CA12CA1CA2CA9
SCHEMBL11879420 0.89 CA12 (0.56) RAD51CA12CA1CA2CA9
SCHEMBL8012728 0.89 RAD51 (0.54) RAD51CA12CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5912221-A POLYMERS FOR INHIBITING DYE DEPOSITION ON FABRICS WITH SURFACTANTS PROCTER & GAMBLE COMPANY (US) 1999-06-15 US disclosed