SCHEMBL846680

SCHEMBL846680

Nc1cc2ccccc2nc1Cl

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.55
ALDH1A1 P00352 5/20 0.52
MAPT P10636 4/20 0.52
HPGD P15428 3/20 0.52
GLA P06280 3/20 0.52
ACHE P22303 1/20 0.52
TDP1 Q9NUW8 1/20 0.52
KDM4E B2RXH2 5/20 0.52
GAA P10253 4/20 0.52
NPC1 O15118 3/20 0.52
POLB P06746 2/20 0.52
RAB9A P51151 2/20 0.52
LMNA P02545 1/20 0.52
PTBP1 P26599 1/20 0.52
RCE1 Q9Y256 1/20 0.52
CASP6 P55212 1/20 0.48
HTR3A P46098 1/20 0.48
MEN1 O00255 2/20 0.46
USP2 O75604 1/20 0.46
CACNA1B Q00975 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4944778 0.86 KMT2A (0.44) KMT2AALDH1A1MAPTHPGDGLA
SCHEMBL244868 0.77 KMT2A (0.59) KMT2AALDH1A1MAPTHPGDGLA
SCHEMBL29911341 0.77 KMT2A (0.59) KMT2AALDH1A1MAPTHPGDGLA
SCHEMBL29454362 0.77 TLR8 (0.57) KMT2AALDH1A1MAPTHPGDGLA
SCHEMBL359102 0.77 TLR8 (0.57) KMT2AALDH1A1MAPTHPGDGLA
Hydrochloric Acid SCHEMBL27365120 0.76 TLR8 (0.55) KMT2AALDH1A1MAPTHPGDGLA
SCHEMBL17993629 0.76 KMT2A (0.57) KMT2AALDH1A1MAPTHPGDGLA
SCHEMBL31278632 0.76 KMT2A (0.57) KMT2AALDH1A1MAPTHPGDGLA
Acridine SCHEMBL10827474 0.75 ALDH1A1 (0.75) KMT2AALDH1A1MAPTHPGDGLA
SCHEMBL3300463 0.74 TLR8 (0.53) KMT2AALDH1A1MAPTHPGDGLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 61 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111909087-A Preparation method of chiral amino chloroquinoline 珠海润都制药股份有限公司 2020-11-10 CN claimed
US-8394828-B2 Quinoline-derived amide modulators of vanilloid VR1 receptor JANSSEN PHARMACEUTICA, NV (BE) 2013-03-12 US claimed
EP-1603883-B1 QUINOLINE-DERIVED AMIDE MODULATORS OF VANILLOID VR1 RECEPTOR JANSSEN PHARMACEUTICA NV (BE) 2012-03-28 EP claimed
US-20080300236-A1 QUINOLINE-DERIVED AMIDE MODULATORS OF VANILLOID VR1 RECEPTOR CODD ELLEN 2008-12-04 US claimed
EP-1603883-A2 QUINOLINE-DERIVED AMIDE MODULATORS OF VANILLOID VR1 RECEPTOR JANSSEN PHARMACEUTICA N.V. (BE) 2005-12-14 EP claimed
US-20040192728-A1 Quinoline-derived amide modulators of vanilloid VR1 receptor JANSSEN PHARMACEUTICA N.V. (BE) 2004-09-30 US claimed
WO-2004069792-A2 QUINOLINE-DERIVED AMIDE MODULATORS OF VANILLOID VR1 RECEPTOR JANSSEN PHARMACEUTICA N.V. (US) 2004-08-19 WO claimed
US-20250090540-A1 PI3K-ALPHA INHIBITORS AND METHODS OF USE THEREOF RELAY THERAPEUTICS, INC. 2025-03-20 US disclosed
CN-119524878-A Disulfide vacancy SV-Bi2S3/SV-ZnIn2S4 heterojunction photocatalyst and preparation method and application thereof 华东师范大学 2025-02-28 CN disclosed
CN-119264200-A Galactose masking aminoquinoline compound and application thereof 厦门大学 2025-01-07 CN disclosed
EP-4399196-A1 PI3K-ALPHA INHIBITORS AND METHODS OF USE THEREOF Relay Therapeutics, Inc. (US) 2024-07-17 EP disclosed
CN-118201896-A PI 3K-alpha inhibitors and methods of use thereof 传达治疗有限公司 2024-06-14 CN disclosed
CN-117504916-A BN-g-C for degrading chloroquine phosphate 3 N 4 /Cs 3 Bi 2 Br 9 Composite photocatalyst and synthesis method thereof 华东师范大学 2024-02-06 CN disclosed
US-20050054640-A1 1-Amino 1H-imidazoquinolines 3M INNOVATIVE PROPERTIES COMPANY 2005-03-10 US disclosed
US-20040192728-A1 Quinoline-derived amide modulators of vanilloid VR1 receptor JANSSEN PHARMACEUTICA N.V. (BE) 2004-09-30 US disclosed
WO-2004080398-A2 1-AMINO 1H-IMIDAZOQUINOLINES 3M INNOVATIVE PROPERTIES COMPANY (US) 2004-09-23 WO disclosed
US-20040176367-A1 1-Amino 1H-imidazoquinolines 3M INNOVATIVE PROPERTIES COMPANY 2004-09-09 US disclosed
WO-2004069792-A2 QUINOLINE-DERIVED AMIDE MODULATORS OF VANILLOID VR1 RECEPTOR JANSSEN PHARMACEUTICA N.V. (US) 2004-08-19 WO disclosed
CN-1063748-C Naphthalene derivatives, process for preparation thereof, and intermediates therefor TANABE SEIYAKU CO (JP) 2001-03-28 CN disclosed
CN-1142497-A Naphthalene derivatives, process for preparation thereof, and intermediates therefor TANABE SEIYAKU CO (JP) 1997-02-12 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040176367-A1 1-Amino 1H-imidazoquinolines IL2, IFNG, IL4I1 KMT2A 2385/4885ALDH1A1 405/4885MAPT 3758/4885
US-20050054640-A1 1-Amino 1H-imidazoquinolines IL2, IFNG, IL4I1 KMT2A 2385/4885ALDH1A1 405/4885MAPT 3758/4885
US-20040192728-A1 Quinoline-derived amide modulators of vanilloid VR1 receptor TRPV1, OPRL1, TRPV2 KMT2A 2415/4885ALDH1A1 1216/4885MAPT 4519/4885
US-20250090540-A1 PI3K-ALPHA INHIBITORS AND METHODS OF USE THEREOF PIK3CA, PIK3CB, PIK3CD KMT2A 2974/4885ALDH1A1 3698/4885MAPT 3881/4885
US-20080300236-A1 QUINOLINE-DERIVED AMIDE MODULATORS OF VANILLOID VR1 RECEPTOR TRPV1, OPRL1, TRPV2 KMT2A 2415/4885ALDH1A1 1216/4885MAPT 4519/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.