SCHEMBL8537398

SCHEMBL8537398

CCCCOC(=O)N(c1ccc(N=C(c2ccccc2)c2ccccc2)cc1)c1ccc(OC)cc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGIR P43119 2/20 0.43
PTGDR Q13258 2/20 0.43
TSHR P16473 2/20 0.40
CES2 O00748 1/20 0.39
CES1 P23141 1/20 0.39
LMNA P02545 2/20 0.38
TP53 P04637 1/20 0.38
TDP1 Q9NUW8 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
CHRM5 P08912 1/20 0.37
CHRM1 P11229 1/20 0.37
CHRM3 P20309 1/20 0.37
KDM4E B2RXH2 1/20 0.37
HPGD P15428 1/20 0.37
TRPM8 Q7Z2W7 1/20 0.37
ALDH1A1 P00352 2/20 0.37
MAPT P10636 2/20 0.37
MEN1 O00255 1/20 0.37
GAA P10253 1/20 0.37
KMT2A Q03164 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7927967 0.81 CES2 (0.41) PTGIRPTGDRTSHRCES2CES1
SCHEMBL29042899 0.78 TSHR (0.54) PTGIRPTGDRTSHRLMNATP53
SCHEMBL6740204 0.77 CYP3A4 (0.52) PTGIRPTGDRTSHRLMNATDP1
SCHEMBL6548684 0.76 NOS3 (0.55) CES2CES1ALDH1A1MAPTMEN1
SCHEMBL6740971 0.73 CYP3A4 (0.54) PTGIRPTGDRTSHRLMNATP53
SCHEMBL29233093 0.72 LMNA (0.55) PTGIRPTGDRTSHRLMNATP53
SCHEMBL19505630 0.70 ESR1 (0.60) CES2CES1ALDH1A1MAPTMEN1
SCHEMBL17017261 0.70 ESR2 (0.66) CES2CES1
SCHEMBL3661310 0.70 KEAP1 (0.49) TSHRLMNATP53KDM4EHPGD
SCHEMBL10689367 0.69 LTB4R2 (0.54) PTGIRPTGDRTSHRLMNAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999028290-A1 SYNTHESIS OF OLIGOARYLAMINES, AND USES AND REAGENTS RELATED THERETO MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 1999-06-10 WO disclosed