SCHEMBL8549494

SCHEMBL8549494

O=C(NCc1ccncc1)[C@@H]1CCCN1CC(=O)C12CC3CC(CC(C3)C1)C2

nearest known ligand 0.56

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.56
CYP17A1 P05093 3/20 0.56
CYP19A1 P11511 3/20 0.56
P2RX7 Q99572 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.48
HSD11B1 P28845 3/20 0.45
SPHK2 Q9NRA0 1/20 0.42
EPHX1 P07099 1/20 0.42
MAPT P10636 1/20 0.42
F2 P00734 1/20 0.42
HPGD P15428 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C9 P11712 1/20 0.41
PKM P14618 1/20 0.41
CYP2C19 P33261 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8544266 0.89 HPGD (0.54) ALDH1A1P2RX7SMN1; SMN2HSD11B1F2
SCHEMBL8549705 0.85 PKM (0.54) ALDH1A1SMN1; SMN2MAPTF2PKM
SCHEMBL8549491 0.83 KMT2A (0.47) ALDH1A1CYP17A1CYP19A1SMN1; SMN2HSD11B1
SCHEMBL8549484 0.83 KMT2A (0.47) ALDH1A1CYP17A1CYP19A1SMN1; SMN2HSD11B1
SCHEMBL8543196 0.83 HSD11B1 (0.62) ALDH1A1P2RX7SMN1; SMN2HSD11B1PKM
SCHEMBL8543051 0.77 RAB9A (0.56) ALDH1A1SMN1; SMN2HPGDCYP2C19
SCHEMBL8546687 0.75 MAPK1 (0.57) ALDH1A1SMN1; SMN2HSD11B1F2CYP3A4
SCHEMBL8543192 0.75 HSD11B1 (0.54) ALDH1A1P2RX7SMN1; SMN2HSD11B1EPHX1
SCHEMBL8548918 0.75 HSD11B1 (0.54) ALDH1A1P2RX7SMN1; SMN2HSD11B1EPHX1
SCHEMBL8544264 0.74 HSD11B1 (0.46) ALDH1A1P2RX7HSD11B1EPHX1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0564924-B1 2-Oxoethyl derivatives as immunosuppressants BAYER AG (US) 1998-09-09 EP claimed
EP-0564924-B1 2-Oxoethyl derivatives as immunosuppressants BAYER AG (US) 1998-09-09 EP disclosed
EP-0564924-A2 2-Oxoethyl derivatives as immunosuppressants Bayer Corporation (US) 1993-10-13 EP disclosed