SCHEMBL8570812

SCHEMBL8570812

COc1ccc(NC(=O)c2ccccc2Cl)cc1C(=O)CCCCCl

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM4 Q14833 7/20 0.54
KMT2A Q03164 3/20 0.53
ALDH1A1 P00352 2/20 0.53
KDM4E B2RXH2 1/20 0.53
SMN1; SMN2 Q16637 4/20 0.53
NPC1 O15118 3/20 0.53
MAPT P10636 3/20 0.53
RAB9A P51151 3/20 0.53
HPGD P15428 1/20 0.53
CYP1A2 P05177 1/20 0.53
CYP3A4 P08684 1/20 0.53
CYP2D6 P10635 1/20 0.53
CYP2C9 P11712 1/20 0.53
CYP2C19 P33261 1/20 0.53
HSD17B10 Q99714 1/20 0.52
HDAC1 Q13547 1/20 0.51
HDAC8 Q9BY41 1/20 0.51
HDAC6 Q9UBN7 1/20 0.51
PNLIP P16233 2/20 0.51
MEN1 O00255 2/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8567801 0.87 KCNK3 (0.55) KMT2AALDH1A1KDM4ESMN1; SMN2NPC1
SCHEMBL8574070 0.85 ALDH1A1 (0.51) KMT2AALDH1A1KDM4EMAPTCYP3A4
SCHEMBL5023609 0.80 PTGS2 (0.72) GRM4KMT2AALDH1A1KDM4ESMN1; SMN2
SCHEMBL195970 0.80 SMN1; SMN2 (0.78) GRM4KMT2AALDH1A1KDM4ESMN1; SMN2
SCHEMBL8809240 0.78 GAA (0.59) ALDH1A1SMN1; SMN2NPC1RAB9AHDAC1
SCHEMBL8569591 0.77 HDAC8 (0.67) KMT2AALDH1A1SMN1; SMN2NPC1RAB9A
SCHEMBL11313551 0.77 KDM4E (0.62) GRM4KMT2AALDH1A1KDM4ESMN1; SMN2
SCHEMBL8570504 0.76 HTR6 (0.52) KMT2AALDH1A1KDM4ESMN1; SMN2HSD17B10
SCHEMBL8571105 0.76 HTR2A (0.55) KMT2AALDH1A1MAPTCYP1A2CYP2C19
SCHEMBL8570818 0.74 NPC1 (0.51) KMT2AALDH1A1KDM4ESMN1; SMN2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5739336-A SELECTIVE 5-HYDROXYTRYPTAMINE-2C RECEPTOR ANTAGONISTS SYNTEX (U.S.A.) INC. (US) 1998-04-14 US disclosed
WO-1997000872-A1 1,3,8-TRIAZA- AND 3,8-DIAZA-1-OXASPIRO(4,5)DECANE DERIVATIVES F.HOFFMANN-LA ROCHE AG (CH) 1997-01-09 WO disclosed