SCHEMBL8630813

SCHEMBL8630813

Cc1cc(Nc2ccccc2C(F)(F)F)c(S(C)(=O)=O)cc1C(=O)Cl

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 1/20 0.50
AKR1C2 P52895 1/20 0.50
TAS2R14 Q9NYV8 3/20 0.43
CYP1A2 P05177 2/20 0.43
CYP2C19 P33261 2/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
TSHR P16473 2/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
ALDH1A1 P00352 5/20 0.42
ALOX12 P18054 3/20 0.42
TP53 P04637 1/20 0.42
BCL2L1 Q07817 1/20 0.42
MCL1 Q07820 1/20 0.42
CNR2 P34972 1/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
HTT P42858 1/20 0.40
PLA2G1B P04054 1/20 0.40
CYP2C9 P11712 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8633397 0.86 AKR1C3 (0.43) AKR1C3AKR1C2TAS2R14CYP1A2CYP2C19
SCHEMBL8631388 0.84 GAA (0.40) ALDH1A1SMN1; SMN2HTT
SCHEMBL7764868 0.84 SLC9A1 (0.56)
SCHEMBL8636232 0.83 PTGS2 (0.40) AKR1C3CYP1A2CYP2C19MEN1KMT2A
SCHEMBL8635463 0.80 AKR1C3 (0.45) AKR1C3AKR1C2MEN1KMT2AALDH1A1
SCHEMBL8634356 0.80 AKR1C3 (0.49) AKR1C3AKR1C2MEN1KMT2AHTT
SCHEMBL8635174 0.80 AKR1C3 (0.49) AKR1C3AKR1C2MEN1KMT2AALDH1A1
SCHEMBL8632107 0.80 AKR1C3 (0.52) AKR1C3AKR1C2
SCHEMBL8633215 0.79 L3MBTL1 (0.42) TAS2R14MEN1KMT2AALDH1A1NPSR1
SCHEMBL8632865 0.76 RORC (0.36) KMT2ACNR2SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5739142-A 4-aminobenzoylguanidine derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1998-04-14 US disclosed