SCHEMBL8743573

SCHEMBL8743573

O=C(O)CNC(=O)c1cccc(Cl)c1Cl

nearest known ligand 0.60

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GPR139 Q6DWJ6 2/20 0.60
P2RX7 Q99572 7/20 0.57
TSHR P16473 1/20 0.56
ERCC5 P28715 1/20 0.54
FEN1 P39748 1/20 0.54
TAS1R3 Q7RTX0 1/20 0.54
TAS1R1 Q7RTX1 1/20 0.54
TAS1R2 Q8TE23 1/20 0.54
TMEM97 Q5BJF2 2/20 0.53
SIGMAR1 Q99720 2/20 0.53
KEAP1 Q14145 1/20 0.51
JAK2 O60674 1/20 0.50
POLB P06746 1/20 0.50
NPC1 O15118 1/20 0.47
RAB9A P51151 1/20 0.47
LMNA P02545 1/20 0.47
HPGD P15428 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2490818 0.86 RAB9A (0.63) GPR139KEAP1POLBNPC1RAB9A
SCHEMBL9491955 0.86 TAS1R3 (0.57) GPR139P2RX7TSHRERCC5FEN1
SCHEMBL23014241 0.84 GPR139 (0.59) GPR139P2RX7TSHRERCC5FEN1
SCHEMBL11570780 0.81 TAS1R3 (0.55) GPR139P2RX7TSHRERCC5FEN1
SCHEMBL4158170 0.81 TAS1R3 (0.64) GPR139P2RX7TSHRERCC5FEN1
SCHEMBL4994139 0.80 ALDH1A1 (0.59) P2RX7FEN1JAK2POLBHPGD
SCHEMBL23014176 0.80 P2RX7 (0.58) GPR139P2RX7TSHRERCC5FEN1
SCHEMBL6292862 0.79 TMEM97 (0.58) GPR139P2RX7TSHRERCC5FEN1
SCHEMBL6292861 0.79 P2RX7 (0.57) GPR139P2RX7TSHRERCC5FEN1
SCHEMBL31448014 0.79 KEAP1 (0.62) TSHRKEAP1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0751929-A1 ANALYSIS METHOD FOR TESTING FOR TRACES OF BETA-AGONISTS AND BETA-ANTAGONISTS UNIVERSITEIT GENT, LABORATORIUM ORGANISCHE CHEMIE, FAKULTEIT LANDBOUWKUNDIGE EN TOEGEPASTE BIOLOGISCHE WETENSCHAPPEN (BE) 1997-01-08 EP disclosed
WO-1995026330-A1 ANALYSIS METHOD FOR TESTING FOR TRACES OF BETA-AGONISTS AND BETA-ANTAGONISTS UNIVERSITEIT GENT, LABORATORIUM ORGANISCHE CHEMIE, FAKULTEIT LANDBOUWKUNDIGE EN TOEGEPASTE BIOLOGISCHE WETENSCHAPPEN (BE) 1995-10-05 WO disclosed