SCHEMBL8774669

SCHEMBL8774669

CCOc1ccc(CCc2cnc(F)c(F)c2)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NQO1 P15559 1/20 0.44
MAPT P10636 1/20 0.43
RAB9A P51151 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
GPR84 Q9NQS5 1/20 0.42
TDP1 Q9NUW8 2/20 0.41
ALDH1A1 P00352 1/20 0.41
TP53 P04637 1/20 0.41
POLB P06746 1/20 0.41
PDGFRB P09619 1/20 0.40
PDGFRA P16234 1/20 0.40
SLC5A1 P13866 1/20 0.40
SLC5A2 P31639 1/20 0.40
SYK P43405 1/20 0.40
MAOB P27338 2/20 0.39
LMNA P02545 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
DHFR P00374 1/20 0.38
SIGMAR1 Q99720 1/20 0.38
TSHR P16473 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8774178 0.88 CYP3A4 (0.43) MAPTRAB9AL3MBTL1ALDH1A1LMNA
SCHEMBL8774716 0.88 LMNA (0.47) MAPTRAB9AL3MBTL1ALDH1A1POLB
SCHEMBL8774858 0.85 MEN1 (0.44) MAPTRAB9AL3MBTL1ALDH1A1LMNA
SCHEMBL8775147 0.83 NPC1 (0.47) MAPTRAB9AGPR84TP53PDGFRB
SCHEMBL8774752 0.83 TAAR1 (0.44) RAB9AL3MBTL1GPR84ALDH1A1TP53
SCHEMBL8774481 0.81 NFKB1 (0.44) MAPTRAB9AL3MBTL1TDP1ALDH1A1
SCHEMBL8110627 0.80 NQO1 (0.50) NQO1GPR84TDP1SLC5A1SLC5A2
SCHEMBL8774132 0.79 NPC1 (0.40) RAB9AL3MBTL1GPR84TP53PDGFRB
SCHEMBL8774337 0.79 RAB9A (0.50) MAPTRAB9AL3MBTL1ALDH1A1TP53
SCHEMBL8774796 0.79 NQO1 (0.41) NQO1GPR84TDP1ALDH1A1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0519370-B1 Heterocyclic derivatives MERCK PATENT GMBH (DE) 1997-11-05 EP disclosed
EP-0519370-A2 Heterocyclic derivatives MERCK PATENT GmbH (DE) 1992-12-23 EP disclosed