SCHEMBL8774752

SCHEMBL8774752

CCc1ccc(CCc2cnc(F)c(F)c2)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 1/20 0.44
L3MBTL1 Q9Y468 2/20 0.38
TP53 P04637 2/20 0.37
NPC1 O15118 1/20 0.37
PKM P14618 1/20 0.37
RAB9A P51151 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
HSD17B10 Q99714 1/20 0.37
GPR84 Q9NQS5 2/20 0.36
LMNA P02545 1/20 0.35
PDGFRB P09619 1/20 0.35
PDGFRA P16234 1/20 0.35
KDM4E B2RXH2 1/20 0.34
HRH3 Q9Y5N1 1/20 0.34
HTR2A P28223 1/20 0.34
KCNH2 Q12809 1/20 0.34
ALDH1A1 P00352 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2D6 P10635 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8774132 0.95 NPC1 (0.40) TAAR1L3MBTL1TP53NPC1PKM
SCHEMBL8775147 0.89 NPC1 (0.47) TP53NPC1PKMRAB9ASMN1; SMN2
SCHEMBL8774481 0.86 NFKB1 (0.44) L3MBTL1TP53NPC1PKMRAB9A
SCHEMBL8774337 0.85 RAB9A (0.50) TAAR1L3MBTL1TP53NPC1PKM
SCHEMBL12188705 0.85 RXRA (0.33) L3MBTL1TP53NPC1PKMRAB9A
SCHEMBL8774239 0.83 HTR2A (0.50) L3MBTL1TP53NPC1RAB9ASMN1; SMN2
SCHEMBL8774669 0.83 NQO1 (0.44) L3MBTL1TP53RAB9ASMN1; SMN2GPR84
SCHEMBL8774784 0.82 RAB9A (0.46) L3MBTL1TP53NPC1PKMRAB9A
SCHEMBL8774178 0.81 CYP3A4 (0.43) L3MBTL1NPC1PKMRAB9ASMN1; SMN2
SCHEMBL8774716 0.81 LMNA (0.47) L3MBTL1NPC1RAB9ASMN1; SMN2HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0519370-B1 Heterocyclic derivatives MERCK PATENT GMBH (DE) 1997-11-05 EP disclosed
EP-0519370-A2 Heterocyclic derivatives MERCK PATENT GmbH (DE) 1992-12-23 EP disclosed