SCHEMBL8870992

SCHEMBL8870992

O=C(Cc1c[nH]c2ccc(F)cc12)N1CCC(n2ccc3c(F)cccc32)CC1

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.47
PTGDR2 Q9Y5Y4 1/20 0.44
SLC6A4 P31645 4/20 0.43
TACR1 P25103 1/20 0.41
TACR3 P29371 1/20 0.41
ICMT O60725 1/20 0.41
ACHE P22303 4/20 0.41
HTR1A P08908 3/20 0.41
HSD11B1 P28845 1/20 0.41
SOS1 Q07889 1/20 0.41
ANO1 Q5XXA6 1/20 0.40
HTR1D P28221 1/20 0.40
HTR1B P28222 1/20 0.40
CDK4 P11802 1/20 0.40
CCND1 P24385 1/20 0.40
MPO P05164 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8871407 0.91 KMT2A (0.48) SLC6A4ACHEHTR1AHTR1DHTR1B
SCHEMBL8871654 0.82 MPO (0.59) SLC6A4HTR1ACDK4CCND1MPO
SCHEMBL8870466 0.80 HTR1A (0.63) SLC6A4HTR1AMPO
SCHEMBL8870996 0.80 TSHR (0.47) TSHRPTGDR2SLC6A4TACR1TACR3
SCHEMBL8557474 0.79 HSD11B1 (0.48) TSHRPTGDR2SLC6A4TACR1TACR3
SCHEMBL8556742 0.77 HSD11B1 (0.61) TSHRSLC6A4HTR1AHSD11B1HTR1D
SCHEMBL9541312 0.74 TSHR (0.60) TSHRPTGDR2SLC6A4ACHEHTR1A
SCHEMBL8870741 0.73 TSHR (0.50) TSHRPTGDR2SLC6A4TACR1TACR3
SCHEMBL8871409 0.71 KMT2A (0.51) SLC6A4ACHEHTR1AHSD11B1MPO
SCHEMBL23244251 0.70 ME2 (0.59) TSHRSLC6A4ACHEHTR1AHTR1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5693655-A 3-indolylpiperidines MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1997-12-02 US disclosed