SCHEMBL8917617

SCHEMBL8917617

CCCCN(CCCC)C(=O)c1ccc(S(=O)(=O)NC(=O)c2cnc(C(=O)NCC(=O)O)c(OC)c2)cc1

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
LIMK1 P53667 1/20 0.42
LIMK2 P53671 1/20 0.42
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA9 Q16790 1/20 0.40
P4HTM Q9NXG6 2/20 0.39
EGLN1 Q9GZT9 4/20 0.39
HDAC1 Q13547 2/20 0.37
HDAC6 Q9UBN7 2/20 0.37
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
LPAR1 Q92633 3/20 0.37
PTGS2 P35354 1/20 0.36
LPAR5 Q9H1C0 1/20 0.36
HDAC3 O15379 1/20 0.36
HDAC2 Q92769 1/20 0.36
HDAC8 Q9BY41 1/20 0.36
SMPD1 P17405 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8916746 0.92 EGLN1 (0.42) LIMK1LIMK2CA1CA2CA9
SCHEMBL8875242 0.91 LIMK1 (0.39) LIMK1LIMK2CA2P4HTMKDM4E
SCHEMBL8874117 0.86 P4HTM (0.38) LIMK1CA2P4HTMKDM4EALDH1A1
SCHEMBL8915935 0.84 PTGS2 (0.51) P4HTMEGLN1PTGS2
SCHEMBL8869660 0.84 P4HTM (0.48) LIMK1LIMK2CA1CA2CA9
SCHEMBL8875238 0.83 MEN1 (0.44) P4HTMSMPD1
SCHEMBL8768258 0.83 CA1 (0.39) LIMK1LIMK2CA1CA2CA9
SCHEMBL8875475 0.83 P4HTM (0.39) P4HTMALDH1A1PTGS2
SCHEMBL8875237 0.82 P4HTM (0.38) P4HTMEGLN1PTGS2
SCHEMBL8917435 0.82 LMNA (0.38) LIMK1LIMK2CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5610172-A Sulfonamidocarbonylpyridine-2-carboxamides and pyridine-n-oxides which are useful as pharmaceuticals HOECHST AKTIENGESELLSCHAFT (DE) 1997-03-11 US disclosed