SCHEMBL8968832

SCHEMBL8968832

CC(C)(C)c1ccc(C#N)cc1NC(=Nc1ccccc1)NC#N

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCC9 O60706 6/20 0.42
KCNJ11 Q14654 6/20 0.42
IMPDH2 P12268 1/20 0.38
KMT2A Q03164 1/20 0.36
CXCR2 P25025 4/20 0.36
CXCR1 P25024 3/20 0.36
P2RX7 Q99572 3/20 0.34
ADRB2 P07550 1/20 0.34
ADRB1 P08588 1/20 0.34
ADRB3 P13945 1/20 0.34
GAA P10253 1/20 0.33
GRIN2D O15399 1/20 0.33
GRIN3B O60391 1/20 0.33
GRIN1 Q05586 1/20 0.33
GRIN2A Q12879 1/20 0.33
GRIN2B Q13224 1/20 0.33
GRIN2C Q14957 1/20 0.33
GRIN3A Q8TCU5 1/20 0.33
SIGMAR1 Q99720 1/20 0.33
NOS3 P29474 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8968206 0.87 ABCC9 (0.42) ABCC9KCNJ11IMPDH2KMT2AP2RX7
SCHEMBL6817607 0.80 CXCR2 (0.53) ABCC9KCNJ11IMPDH2CXCR2CXCR1
SCHEMBL8968827 0.77 CXCR2 (0.44) ABCC9KCNJ11KMT2ACXCR2CXCR1
SCHEMBL8968824 0.77 CXCR2 (0.44) ABCC9KCNJ11KMT2ACXCR2CXCR1
SCHEMBL6818380 0.74 IMPDH2 (0.41) ABCC9KCNJ11IMPDH2CXCR2CXCR1
SCHEMBL8968160 0.74 CXCR2 (0.65) KMT2ACXCR2CXCR1GAA
SCHEMBL8968189 0.71 ALDH1A1 (0.43) KMT2ACXCR2CXCR1GAA
SCHEMBL8968209 0.71 KMT2A (0.36) KMT2ACXCR2CXCR1GAA
SCHEMBL9235204 0.71 KMT2A (0.36) KMT2ACXCR2CXCR1GAA
SCHEMBL8968156 0.70 GAA (0.49) CXCR2CXCR1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0656350-A1 Biaryl urea and related compounds BRISTOL-MYERS SQUIBB COMPANY (US) 1995-06-07 EP claimed
US-5547966-A Aryl urea and related compounds BRISTOL-MYERS SQUIBB COMPANY (US) 1996-08-20 US disclosed
EP-0656350-A1 Biaryl urea and related compounds BRISTOL-MYERS SQUIBB COMPANY (US) 1995-06-07 EP disclosed