SCHEMBL8997593

SCHEMBL8997593

COC(=O)O[C@]1(NC(=O)OC(C)(C)C)CCc2cccc(Oc3ccccc3CNC(=O)[C@H](C)NC(=O)CCNC(=O)OCc3ccccc3)c2C1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.35
CYP3A4 P08684 3/20 0.35
CYP2C9 P11712 3/20 0.35
CYP2C19 P33261 3/20 0.35
CYP1A2 P05177 2/20 0.35
HPGD P15428 1/20 0.35
HSD17B10 Q99714 1/20 0.35
SYK P43405 1/20 0.35
MAPT P10636 3/20 0.34
LMNA P02545 3/20 0.34
REN P00797 1/20 0.34
KLK7 P49862 2/20 0.33
KLK5 Q9Y337 2/20 0.33
CYP2D6 P10635 2/20 0.33
TSHR P16473 1/20 0.33
HTT P42858 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
ACHE P22303 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8997600 0.89 SYK (0.40) ALDH1A1CYP3A4CYP2C9CYP2C19CYP1A2
SCHEMBL8997611 0.81 RPS6KA1 (0.34) ALDH1A1CYP3A4HPGDHSD17B10PSMB5
SCHEMBL8997612 0.79 SYK (0.41) ALDH1A1CYP3A4CYP2C9CYP2C19CYP1A2
SCHEMBL8575729 0.79 CA1 (0.39) ALDH1A1CYP3A4SYKMAPTKLK7
SCHEMBL8567143 0.79 CA1 (0.39) ALDH1A1CYP3A4SYKMAPTKLK7
SCHEMBL8997594 0.78 SYK (0.40) ALDH1A1CYP3A4CYP2C9CYP2C19CYP1A2
SCHEMBL8581093 0.78 GHSR (0.40) SYKMAPTCA1CA2ACHE
SCHEMBL8997625 0.77 GHSR (0.37) CYP2C9CYP1A2MAPTLMNASMN1; SMN2
SCHEMBL8997648 0.76 SYK (0.38) SYKKLK7KLK5CA1CA2
SCHEMBL8997603 0.76 SYK (0.38) CYP3A4CYP2C9CYP2C19CYP1A2SYK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0729972-A1 Peptide derivatives of tetrahydronaphthalene F. HOFFMANN-LA ROCHE AG (CH) 1996-09-04 EP disclosed