SCHEMBL9032018

SCHEMBL9032018

COc1ccc(-c2ccncc2)cc1C(N)c1occ2ccccc12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHFR P00374 3/20 0.39
MAPT P10636 3/20 0.36
SMN1; SMN2 Q16637 3/20 0.36
NPC1 O15118 2/20 0.36
KDM4E B2RXH2 2/20 0.36
ALDH1A1 P00352 2/20 0.36
TLR9 Q9NR96 2/20 0.36
USP2 O75604 1/20 0.36
LMNA P02545 1/20 0.36
TSHR P16473 1/20 0.36
HSD17B10 Q99714 1/20 0.36
TLR8 Q9NR97 1/20 0.36
TLR7 Q9NYK1 1/20 0.36
ABCB1 P08183 1/20 0.35
ABCG2 Q9UNQ0 1/20 0.35
S1PR1 P21453 1/20 0.35
S1PR3 Q99500 1/20 0.35
PDE4A P27815 1/20 0.35
HPGD P15428 1/20 0.35
CYP17A1 P05093 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9026336 0.88 CYP11B2 (0.47) MAPTSMN1; SMN2NPC1KDM4EALDH1A1
SCHEMBL9025514 0.85 PDE4A (0.39) MAPTSMN1; SMN2NPC1KDM4EALDH1A1
SCHEMBL9025454 0.82 CA12 (0.34) MAPTSMN1; SMN2KDM4EALDH1A1LMNA
SCHEMBL9026859 0.81 ADRA2A (0.45) MAPTNPC1KDM4EALDH1A1TSHR
SCHEMBL9025089 0.81 KDM4E (0.41) MAPTSMN1; SMN2NPC1KDM4EALDH1A1
SCHEMBL9025520 0.81 METAP2 (0.38) MAPTKDM4EALDH1A1LMNATSHR
SCHEMBL9024896 0.80 MYB (0.36) MAPTNPC1LMNATSHRRAB9A
SCHEMBL9216019 0.80 NQO1 (0.36) MAPT
SCHEMBL9025568 0.80 METAP2 (0.39) MAPTNPC1KDM4EALDH1A1RAB9A
SCHEMBL9026008 0.80 PKM (0.38) MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0711290-A1 METHYLGUANIDINE DERIVATIVES, METHODS FOR PREPARING SAME AND COMPOSITIONS CONTAINING SAID DERIVATIVES SANOFI (FR) 1996-05-15 EP disclosed
WO-1995004052-A1 METHYLGUANIDINE DERIVATIVES, METHODS FOR PREPARING SAME AND COMPOSITIONS CONTAINING SAID DERIVATIVES SANOFI (FR) 1995-02-09 WO disclosed