SCHEMBL907784

SCHEMBL907784

CCOc1c[c]cc(OCC)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NQO1 P15559 1/20 0.52
TSHR P16473 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
TP53 P04637 1/20 0.41
CYP3A4 P08684 1/20 0.41
ESR1 P03372 2/20 0.39
AHR P35869 1/20 0.39
LTA4H P09960 2/20 0.39
MEN1 O00255 1/20 0.38
NPC1 O15118 1/20 0.38
KMT2A Q03164 1/20 0.38
APOBEC3G Q9HC16 1/20 0.38
ALDH1A1 P00352 2/20 0.36
MAPT P10636 1/20 0.36
ESR2 Q92731 1/20 0.36
HSD17B10 Q99714 1/20 0.36
HPGD P15428 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2D6 P10635 1/20 0.36
MAPK1 P28482 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL499727 0.91 ESR1 (0.47) NQO1TSHRTDP1TP53CYP3A4
SCHEMBL9797716 0.89 NQO1 (0.42) NQO1TSHRTDP1TP53CYP3A4
SCHEMBL16952712 0.87 NQO1 (0.46) NQO1TSHRTDP1CYP3A4AHR
SCHEMBL4880339 0.85 NQO1 (0.44) NQO1TSHRTDP1TP53CYP3A4
SCHEMBL5740806 0.85 NQO1 (0.44) NQO1TSHRTDP1TP53CYP3A4
SCHEMBL16953037 0.85 NQO1 (0.39) NQO1TSHRTDP1TP53CYP3A4
SCHEMBL16960727 0.85 NQO1 (0.39) NQO1TSHRTDP1TP53CYP3A4
SCHEMBL16952562 0.85 NQO1 (0.39) NQO1TSHRTDP1TP53CYP3A4
SCHEMBL457601 0.84 NQO1 (0.42) NQO1TSHRTDP1TP53CYP3A4
SCHEMBL10858288 0.84 TP53 (0.53) NQO1TSHRTDP1TP53CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 390 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3324974-B1 COMPOUNDS, COMPOSITIONS, METHODS FOR TREATING DISEASES, AND METHODS FOR PREPARING COMPOUNDS UNIV LOUISVILLE RES FOUND INC (US) 2022-06-08 EP claimed
US-11312690-B2 Compounds, compositions, methods for treating diseases, and methods for preparing compounds UNIVERSITY OF LOUSVILLE RESEARCH FOUNDATION, INC. (US) 2022-04-26 US claimed
US-11208379-B2 Compounds, compositions, methods for treating diseases, and methods for preparing compounds UNIVERSITY OF LOUISVILLE RESEARCH FOUNDATION, INC. (US) 2021-12-28 US claimed
US-20210355064-A1 METHODS RELATED TO CARBON DIOXIDE UNIVERSITY OF LOUISVILLE RESEARCH FOUNDATION, INC. (US) 2021-11-18 US claimed
CN-113444125-A Novel phosphoramidite ligand, preparation method thereof and application thereof in asymmetric carbonylation reaction 西北大学 2021-09-28 CN claimed
US-11078148-B2 Methods for the reduction of carbon dioxide UNIVERSITY OF LOUISVILLE RESEARCH FOUNDATION, INC. (US) 2021-08-03 US claimed
US-20210138117-A1 COMPOUNDS AND MATRICES FOR USE IN BONE GROWTH AND REPAIR HUMAN BIOMOLECULAR RESEARCH INSTITUTE (US) 2021-05-13 US claimed
EP-3038621-B1 COMPOUNDS AND MATRICES FOR USE IN BONE GROWTH AND REPAIR HUMAN BIOMOLECULAR RES INSTITUTE (US) 2020-12-02 EP claimed
US-20200277248-A1 METHODS FOR THE REDUCTION OF CARBON DIOXIDE UNIVERSITY OF LOUISVILLE RESEARCH FOUNDATION, INC. (US) 2020-09-03 US claimed
US-20200079742-A1 COMPOUNDS, COMPOSITIONS, METHODS FOR TREATING DISEASES, AND METHODS FOR PREPARING COMPOUNDS UNIVERSITY OF LOUSVILLE RESEARCH FOUNDATION, INC. (US) 2020-03-12 US claimed
US-20080223444-A1 Perylene Charge-Transport Materials, Methods of Fabrication Thereof, and Methods of Use Thereof GEORGIA TECH RESEARCH CORPORATION 2008-09-18 US claimed
WO-2006127024-A1 REAGENTS AND METHODS FOR LABELING TERMINAL OLEFINS EISAI CO. LTD. (JP) 2006-11-30 WO claimed
WO-2006093965-A2 CORONENE CHARGE-TRANSPORT MATERIALS, METHODS OF FABRICATION THEREOF, AND METHODS OF USE THEREOF GEORGIA TECH RESEARCH CORPORATION (US) 2006-09-08 WO claimed
US-20060045846-A1 Reagents and methods for labeling terminal olefins EISAI R&D MANAGEMENT CO., LTD. (JP) 2006-03-02 US claimed
WO-2005124453-A2 PERYLENE CHARGE-TRANSPORT MATERIALS, METHODS OF FABRICATION THEREOF, AND METHODS OF USE THEREOF GEORGIA TECH RESEARCH CORPORATION (US) 2005-12-29 WO claimed
US-6124478-A Methods of using 1,2-dioxetanes and kits therefore TROPIX, INC. (US) 2000-09-26 US claimed
EP-0536896-B1 Imidazolidyl macrolides having immunosuppressive activity MERCK & CO INC (US) 1997-12-17 EP claimed
US-5247076-A IMIDAZOLIDYL MACROLIDES HAVING IMMUNOSUPPRESSIVE ACTIVITY MERCK & CO., INC. (US) 1993-09-21 US claimed
EP-0536896-A1 Imidazolidyl macrolides having immunosuppressive activity MERCK & CO. INC. (US) 1993-04-14 EP claimed
WO-1993005059-A1 IMIDAZOLIDYL MACROLIDES MERCK & CO., INC. (US) 1993-03-18 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (9 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200277248-A1 METHODS FOR THE REDUCTION OF CARBON DIOXIDE CA5A, CA5B, FTO NQO1 170/4885TSHR 3993/4885TDP1 3559/4885
US-20210355064-A1 METHODS RELATED TO CARBON DIOXIDE CA1, CA5A, CA9 NQO1 460/4885TSHR 4033/4885TDP1 3599/4885
US-20210138117-A1 COMPOUNDS AND MATRICES FOR USE IN BONE GROWTH AND REPAIR BMP2, BMP4, BMP6 NQO1 2074/4885TSHR 2887/4885TDP1 4775/4885
US-11208379-B2 Compounds, compositions, methods for treating diseases, and methods for preparing compounds VHL, KRAS, C5 NQO1 152/4885TSHR 4685/4885TDP1 2341/4885
US-11078148-B2 Methods for the reduction of carbon dioxide CA5A, CA5B, FTO NQO1 170/4885TSHR 3993/4885TDP1 3559/4885
US-20080223444-A1 Perylene Charge-Transport Materials, Methods of Fabrication Thereof, and Methods of Use Thereof SLC43A1, SLC3A2, SLC16A3 NQO1 1178/4885TSHR 4842/4885TDP1 924/4885
US-20060045846-A1 Reagents and methods for labeling terminal olefins EEF2, RNF168, REL NQO1 1800/4885TSHR 469/4885TDP1 3131/4885
US-20200079742-A1 COMPOUNDS, COMPOSITIONS, METHODS FOR TREATING DISEASES, AND METHODS FOR PREPARING COMPOUNDS VHL, C5, KRAS NQO1 157/4885TSHR 4651/4885TDP1 2610/4885
US-11312690-B2 Compounds, compositions, methods for treating diseases, and methods for preparing compounds VHL, C5, KRAS NQO1 157/4885TSHR 4651/4885TDP1 2610/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.