SCHEMBL9084422

SCHEMBL9084422

O=C=C1CC(N2CCCC2=O)CCN1OCc1ccccc1

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 1/20 0.36
LTA4H P09960 4/20 0.36
KCNH2 Q12809 2/20 0.36
ALDH1A1 P00352 3/20 0.36
THRB P10828 1/20 0.36
MGLL Q99685 1/20 0.34
RORC P51449 1/20 0.34
CYP2D6 P10635 1/20 0.34
HRH1 P35367 1/20 0.34
PSEN1 P49768 1/20 0.33
PSEN2 P49810 1/20 0.33
APH1B Q8WW43 1/20 0.33
NCSTN Q92542 1/20 0.33
APH1A Q96BI3 1/20 0.33
PSENEN Q9NZ42 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9082309 0.97 LTA4H (0.38) CASP1LTA4HKCNH2ALDH1A1THRB
SCHEMBL9115852 0.85 FKBP1A (0.33) ALDH1A1
SCHEMBL5871698 0.76 ALDH1A1 (0.41) CASP1ALDH1A1
SCHEMBL7448545 0.74 SMN1; SMN2 (0.53) LTA4HALDH1A1
SCHEMBL6947156 0.72 CASP1 (0.53) CASP1ALDH1A1
SCHEMBL9204131 0.71 CTSL (0.36) ALDH1A1
SCHEMBL1286296 0.71 ALDH1A1 (0.41) ALDH1A1
SCHEMBL9796122 0.70 ALDH1A1 (0.38) ALDH1A1
SCHEMBL6969799 0.70 SMN1; SMN2 (0.61) CYP2D6
SCHEMBL4585565 0.69 LTA4H (0.60) LTA4HKCNH2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5559131-A ANTAGONISTS OF TACHYKININS AT THE NEUROKININ 2 RECEPTOR, ANTIASTHMA ZENECA LIMITED (GB) 1996-09-24 US disclosed
EP-0667858-A1 4-CARBOXOAMIDO PIPERIDINE DERIVATIVES, INTERMEDIATES AND USE AS NEUROKININ ANTAGONISTS ZENECA LIMITED (GB) 1995-08-23 EP disclosed