SCHEMBL9117010

SCHEMBL9117010

COC(=O)C1(C(=O)OC)C=C(c2ccc(C(F)(F)F)cn2)C(c2ccccc2S(N)(=O)=O)=C1

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 1/20 0.39
F10 P00742 4/20 0.38
PTGES2 Q9H7Z7 3/20 0.38
HCRTR1 O43613 2/20 0.37
HCRTR2 O43614 2/20 0.37
CCR6 P51684 1/20 0.36
KLK1 P06870 1/20 0.36
ALOX5AP P20292 3/20 0.36
FEN1 P39748 3/20 0.36
CA1 P00915 2/20 0.35
CA2 P00918 2/20 0.35
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
CA5A P35218 1/20 0.35
CA9 Q16790 1/20 0.35
TRPV1 Q8NER1 1/20 0.35
P2RY1 P47900 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8974585 0.82 KIF11 (0.46) KIF11CCR6CA1CA2CA9
SCHEMBL8973879 0.78 KIF11 (0.45) KIF11CA1CA2CA9
SCHEMBL8974421 0.78 PTGS2 (0.43) KIF11
SCHEMBL9117008 0.78 HSD11B1 (0.41) KIF11PTGES2NPC1RAB9A
SCHEMBL6883474 0.78 KIF11 (0.50) KIF11PTGES2HCRTR1HCRTR2ALOX5AP
SCHEMBL8974117 0.74 PTGS2 (0.40)
SCHEMBL8973763 0.70 POLB (0.41) KIF11CA1CA2CA9
SCHEMBL8973781 0.69 KIF11 (0.59) KIF11CA1CA2CA9
SCHEMBL8974757 0.68 CA2 (0.41) CA1CA2CA5ACA9
SCHEMBL8974407 0.68 PTGS2 (0.41) CA1CA2CA5ACA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1995030656-A1 SUBSTITUTED CYCLOPENTADIENYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1995-11-16 WO disclosed