SCHEMBL932791

SCHEMBL932791

CCCCC1=C(O)C(=O)C=CC1=O

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 17/20 0.51
MPEG1 Q2M385 11/20 0.51
XIAP P98170 3/20 0.51
GPR84 Q9NQS5 2/20 0.51
KDM4E B2RXH2 1/20 0.51
MEN1 O00255 1/20 0.51
PTGES O14684 1/20 0.51
USP2 O75604 1/20 0.51
ALDH1A1 P00352 1/20 0.51
TP53 P04637 1/20 0.51
CYP2D6 P10635 1/20 0.51
MAPT P10636 1/20 0.51
CYP2C9 P11712 1/20 0.51
HPGD P15428 1/20 0.51
ALOX15 P16050 1/20 0.51
ALOX12 P18054 1/20 0.51
MAPK1 P28482 1/20 0.51
CYP2C19 P33261 1/20 0.51
KMT2A Q03164 1/20 0.51
KAT2B Q92831 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27904845 0.92 ALOX5 (0.62) ALOX5MPEG1XIAPGPR84KDM4E
SCHEMBL5554116 0.92 ALOX5 (0.62) ALOX5MPEG1XIAPGPR84KDM4E
SCHEMBL7866839 0.84 ACHE (0.47) ALOX5MPEG1XIAPGPR84KDM4E
Butylated Hydroxytoluene SCHEMBL9706618 0.81 SMN1; SMN2 (0.49) ALOX5MPEG1XIAPGPR84KDM4E
SCHEMBL10772074 0.78 XIAP (0.54) ALOX5MPEG1XIAPGPR84KDM4E
SCHEMBL28655350 0.78 ACHE (0.55) ALOX5MPEG1XIAPGPR84KDM4E
SCHEMBL27487222 0.75 ACHE (0.40) ALOX5MPEG1XIAPGPR84KDM4E
SCHEMBL1020312 0.75 ALOX5 (0.65) ALOX5MPEG1XIAPGPR84KDM4E
SCHEMBL19840669 0.75 ACHE (0.37) ALOX5MPEG1XIAPGPR84KDM4E
Hydrochloric Acid SCHEMBL28922225 0.74 ACHE (0.57) ALOX5MPEG1XIAPGPR84KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 207 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230310413-A1 PHARMACEUTICAL FORMULATIONS COMPRISING A MALT1 INHIBITOR AND A MIXTURE OF POLYETHYLENE GLYCOL WITH A FATTY ACID JANSSEN PHARMACEUTICA NV (BE) 2023-10-05 US claimed
US-20230301924-A1 PHARMACEUTICAL FORMULATION Janssen Pharmaceuticals, Inc. 2023-09-28 US claimed
EP-4240334-A1 PHARMACEUTICAL FORMULATION Janssen Pharmaceuticals, Inc. (US) 2023-09-13 EP claimed
EP-4199911-A1 PHARMACEUTICAL FORMULATIONS COMPRISING A MALT1 INHIBITOR AND A MIXTURE OF POLYETHYLENE GLYCOL WITH A FATTY ACID JANSSEN Pharmaceutica NV (BE) 2023-06-28 EP claimed
US-20220175760-A1 PHARMACEUTICAL FORMULATIONS JANSSEN PHARMACEUTICA NV (BE) 2022-06-09 US claimed
WO-2022094817-A1 PHARMACEUTICAL FORMULATION Janssen Pharmaceuticals, Inc. (US) 2022-05-12 WO claimed
WO-2022095912-A1 PHARMACEUTICAL FORMULATION Janssen Pharmaceuticals, Inc. (US) 2022-05-12 WO claimed
WO-2022037661-A1 PHARMACEUTICAL FORMULATIONS COMPRISING A MALT1 INHIBITOR AND A MIXTURE OF POLYETHYLENE GLYCOL WITH A FATTY ACID JANSSEN PHARMACEUTICA NV (BE) 2022-02-24 WO claimed
EP-3927324-A1 PHARMACEUTICAL FORMULATIONS Janssen Pharmaceutica NV (BE) 2021-12-29 EP claimed
US-11191276-B2 Solid formulations suitable for oilfield applications RHODIA OPERATIONS (FR) 2021-12-07 US claimed
US-5650185-A FOOD FLAVORS FOR OILS ACH FOOD COMPANIES, INC. 1997-07-22 US claimed
EP-0607272-B1 NON-AEROSOL, UNIFORM SPRAY DISPERSION SYSTEM FOR OIL-BASED PRODUCTS PAUL LEONARD (US) 1997-03-19 EP claimed
US-5455055-A A food dispenser comprising a housing for holding the food product, a high compression pump to distribute repeatedly, consistently ACH FOOD COMPANIES, INC. 1995-10-03 US claimed
EP-0607272-A4 NON-AEROSOL, UNIFORM SPRAY DISPERSION SYSTEM FOR OIL-BASED PRODUCTS. STOLTZ EDWIN I (US) 1995-02-22 EP claimed
EP-0607272-A1 NON-AEROSOL, UNIFORM SPRAY DISPERSION SYSTEM FOR OIL-BASED PRODUCTS. STOLTZ EDWIN I (US) 1994-07-27 EP claimed
WO-1993006749-A1 NON-AEROSOL, UNIFORM SPRAY DISPERSION SYSTEM FOR OIL-BASED PRODUCTS STOLTZ EDWIN I (US) 1993-04-15 WO claimed
EP-0202512-B1 NICOTINE DISPENSER WITH POLYMERIC RESERVOIR OF NICOTINE Kabi Pharmacia AB (SE) 1992-06-17 EP claimed
US-4761296-A DEFATTING AND IMPREGNATION WITH VEGETABLE OILS NABISCO BRANDS, INC. (US) 1988-08-02 US claimed
US-4736755-A POLYOLEFINS OR POLYOLEFINDIENES, ESPECIALLY POLYETHYLENE AND POLYPROPYLENE ADVANCED TOBACCO PRODUCTS (US) 1988-04-12 US claimed
EP-0169088-A2 Crackers having stabilized sunflower seeds NABISCO BRANDS, Inc. (US) 1986-01-22 EP claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230310413-A1 PHARMACEUTICAL FORMULATIONS COMPRISING A MALT1 INHIBITOR AND A MIXTURE OF POLYETHYLENE GLYCOL WITH A FATTY ACID MALT1, MGAM, MGLL ALOX5 429/4885MPEG1 193/4885XIAP 588/4885
US-20230301924-A1 PHARMACEUTICAL FORMULATION TTPA, PTGES, HMGCR ALOX5 318/4885MPEG1 1157/4885XIAP 2807/4885
US-20220175760-A1 PHARMACEUTICAL FORMULATIONS TREH, F12, CEL ALOX5 1440/4885MPEG1 2689/4885XIAP 2491/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.