SCHEMBL93351

SCHEMBL93351

O=S(=O)([O-])c1nc2c(ccc3c(-c4ccccc4)ccnc32)c(-c2ccccc2)c1S(=O)(=O)[O-].[Na+].[Na+]

nearest known ligand 0.37

Known targets — ChEMBL curated mechanism

ABCC8ACEADORA1ADORA2AADORA2BADORA3ALDH5A1ALOX5ALOX5APATP4AATP4BBRAFCA1CA12CA2CA4CYSLTR1DHFRDPEP1EDNRAEDNRBESR2F10FDPSFGF1GABBR1GABBR2GABRA1GABRA2GABRA3GABRA4GABRA5GABRA6GABRB1GABRB2GABRB3GABRDGABREGABRG1GABRG2GABRG3GABRPGABRQGARTGNRHRGSC1HMGCRIMPDH1IMPDH2KCNJ11LY96NOD2NR3C1NS3NS4ANS5bP2RY1P2RY12P2RY2P2RY4P2RY6PBP2XPDE3APDE3BPDE4APDE4BPDE4CPDE4DPDK1PDK2PDK3PDK4PPARGPPATPTGIRPTGS1PTGS2RAF1RYR1RYR3SCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASERPINC1SLC12A1SLC12A3SYKTHRATHRBTLR3TLR4TLR9TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYMSVKORC1XDHblablaIMP-1blaOXA-33blaOXA-58blaT-3blaT-4blaT-5blaT-6dacAdacBdacCfolAfolPfolP1ftsIfusAgaggyrAgyrBmecAmrcAmrcBmrdApbp1apbp1bpbp2pbp2apbp2bpbp3pbp4pbpApbpBpbpCpbpFpolponBrplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpoArpoBrpoCrpoZrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of None. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN5A known ✓ Q14524 1/20 0.30
SCN9A known ✓ Q15858 1/20 0.30
CKS1B P61024 7/20 0.37
SKP2 Q13309 7/20 0.37
GLO1 Q04760 2/20 0.37
TOP2A P11388 1/20 0.37
NR1H2 P55055 4/20 0.33
NR1H3 Q13133 4/20 0.33
MMP2 P08253 1/20 0.33
IKBKB O14920 1/20 0.33
CHUK O15111 1/20 0.33
DAPK3 O43293 1/20 0.33
JAK2 O60674 1/20 0.33
PRKD3 O94806 1/20 0.33
MAP4K4 O95819 1/20 0.33
PAK4 O96013 1/20 0.33
CSF1R P07333 1/20 0.33
RET P07949 1/20 0.33
IGF1R P08069 1/20 0.33
FGFR1 P11362 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30479688 0.99 CKS1B (0.36) CKS1BSKP2GLO1TOP2ANR1H2
SCHEMBL29026619 0.99 CKS1B (0.36) CKS1BSKP2GLO1TOP2ANR1H2
SCHEMBL769956 0.99 CKS1B (0.36) CKS1BSKP2GLO1TOP2ANR1H2
SCHEMBL2424416 0.99 CKS1B (0.36) CKS1BSKP2GLO1TOP2ANR1H2
SCHEMBL3941509 0.98 CKS1B (0.37) CKS1BSKP2GLO1TOP2ANR1H2
SCHEMBL8775544 0.98 CKS1B (0.37) CKS1BSKP2GLO1TOP2ANR1H2
SCHEMBL3960976 0.98 CKS1B (0.37) CKS1BSKP2GLO1TOP2ANR1H2
SCHEMBL3964610 0.96 CKS1B (0.36) CKS1BSKP2GLO1TOP2ANR1H2
Dipyridyl SCHEMBL17766514 0.93 GLO1 (0.35) CKS1BSKP2GLO1TOP2ANR1H2
SCHEMBL15570898 0.84 TOP2A (0.36) CKS1BSKP2GLO1TOP2ANR1H2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 363 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116949435-A Electroless copper plating solution and method for preparing nano-bicrystal copper metal layer by electroless plating 台湾上村股份有限公司 2023-10-27 CN claimed
US-20230272469-A1 PROTECTIVE SURFACE COATINGS FOR FLOW CELLS ILLUMINA CAMBRIDGE LIMITED (GB) 2023-08-31 US claimed
US-11667969-B2 Protective surface coatings for flow cells ILLUMINA, INC. (US) 2023-06-06 US claimed
CN-115916967-A Production of nucleic acids having modified bases using recombinant terminal deoxynucleotidyl transferases 伊鲁米纳公司 2023-04-04 CN claimed
WO-2023043974-A1 USE OF FLUORESCENT TRACERS TO MONITOR NUTRIENT CONCENTRATIONS IN SOLUTION FEHR SOLUTIONS, LLC (US) 2023-03-23 WO claimed
CN-109689216-B Protective surface coating for flow cell 伊鲁米那股份有限公司 2022-04-05 CN claimed
CN-110075930-B Photocatalytic system with photoresponse switch and self-indicating property as well as preparation method and application 华东师范大学 2020-11-20 CN claimed
CN-109206617-B Method for resolving racemic compound by fractional crystallization 北京大学 2020-04-24 CN claimed
EP-3621735-A1 PROTECTIVE SURFACE COATINGS FOR FLOW CELLS Illumina, Inc. (US) 2020-03-18 EP claimed
CN-110100009-A The chemical connection process of nucleic acid 伊鲁米那股份有限公司 2019-08-06 CN claimed
WO-2003082450-A1 METHOD OF MONITORING MEMBRANE SEPARATION PROCESSES NALCO COMPANY (US) 2003-10-09 WO claimed
WO-2003082447-A1 METHOD OF MONITORING MEMBRANE SEPARATION PROCESSES NALCO COMPANY (US) 2003-10-09 WO claimed
US-20030183575-A1 METHOD OF MONITORING MEMBRANE SEPARATION PROCESSES ECOLAB USA INC. 2003-10-02 US claimed
US-6472219-B1 CONCENTRATION OF TREATMENT PRODUCTS APPLIED TO CUT FLOWER WATER, I.E. IN ORDER TO PREVENT LEAF YELLOWING, ETC. DETERMINED USING FLUOROESCENT INDICATOR ONDEO NALCO COMPANY 2002-10-29 US claimed
WO-2002017717-A1 USE OF TRACERS TO MONITOR APPLICATION OF TREATMENT PRODUCTS TO CUT FLOWERS ONDEO NALCO COMPANY (US) 2002-03-07 WO claimed
EP-0892865-A1 METHOD FOR BLEACHING OF LIGNOCELLULOSIC FIBERS Jaschinski, Thomas (DE) 1999-01-27 EP claimed
WO-1997039179-A1 METHOD FOR BLEACHING OF LIGNOCELLULOSIC FIBERS JASCHINSKI THOMAS (DE) 1997-10-23 WO claimed
EP-0170414-B1 PROCESS FOR TREATING METAL SURFACE Hitachi Chemical Co., Ltd. (JP) 1991-04-17 EP claimed
US-4643793-A WITH MIXTURE OF COPPER COMPOUND, COMPLEXING AGENT, REDUCING AGENT, AND PH ADJUSTER IN PRESENCE OF NITROGEN HETEROCYCLE COMPOUND HITACHI CHEMICAL COMPANY, LTD. (JP) 1987-02-17 US claimed
EP-0170414-A2 Process for treating metal surface Hitachi Chemical Co., Ltd. (JP) 1986-02-05 EP claimed