SCHEMBL9429617

SCHEMBL9429617

Cn1c(N2CCN(CCCC(=O)c3ccc(F)cc3)CC2)cc(=O)n(C)c1=O

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.62
DRD2 P14416 8/20 0.60
DRD4 P21917 8/20 0.60
DRD3 P35462 8/20 0.60
HTR1A P08908 6/20 0.58
HTR2A P28223 5/20 0.58
HTR2C P28335 5/20 0.58
HRH1 P35367 3/20 0.58
ADRA2C P18825 1/20 0.58
ALDH1A1 P00352 1/20 0.57
POLB P06746 1/20 0.57
DRD1 P21728 2/20 0.57
MEN1 O00255 1/20 0.57
CHRM2 P08172 1/20 0.57
ADRA2A P08913 1/20 0.57
ADRA1A P35348 1/20 0.57
OPRM1 P35372 1/20 0.57
KMT2A Q03164 1/20 0.57
KCNH2 Q12809 1/20 0.57
HRH3 Q9Y5N1 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9429271 0.99 TSHR (0.65) TSHRDRD2DRD4DRD3HTR1A
SCHEMBL9429593 0.81 SOD1 (0.57) TSHRDRD2DRD4DRD3HTR1A
SCHEMBL9429398 0.81 HTR1A (0.56) HTR1AHRH1ALDH1A1KMT2A
SCHEMBL9428233 0.81 CACNA1G (0.57) HTR1AALDH1A1HTR7LMNA
Hydrochloric Acid SCHEMBL9428830 0.80 ALDH1A1 (0.56) HTR1AHRH1ALDH1A1KMT2A
SCHEMBL9428373 0.80 DRD2 (0.58) DRD2DRD3HTR1AHTR2AHRH1
Hydrochloric Acid SCHEMBL9428467 0.79 DRD2 (0.57) DRD2DRD3HTR1AHTR2AHRH1
SCHEMBL11832182 0.79 DRD2 (0.88) TSHRDRD2DRD4DRD3HTR1A
SCHEMBL16986166 0.79 TSHR (0.97) TSHRDRD2DRD4DRD3HTR1A
SCHEMBL9428377 0.78 CCR5 (0.44) HRH1ALDH1A1MEN1ADRA1AKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5332739-A Pyrimidinedione derivatives and antiarrhythmic agents containing same MITSUI TOATSU CHEMICALS, INCORPORATED (JP) 1994-07-26 US disclosed
EP-0454498-A2 Pyrimidinedione derivatives and antiarrhythmic agents containing same MITSUI TOATSU CHEMICALS, Inc. (JP) 1991-10-30 EP disclosed