SCHEMBL9535482

SCHEMBL9535482

Cc1nc2n(c(=O)c1CCN1CCC(Cc3nc4ccccc4n3Cc3cccs3)CC1)CCCC2

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 12/20 0.54
HTR2A P28223 12/20 0.54
HTR1A P08908 11/20 0.54
KCNH2 Q12809 4/20 0.48
HTR2C P28335 3/20 0.48
ADRA1A P35348 3/20 0.48
HRH1 P35367 3/20 0.48
TSHR P16473 2/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
SLC22A2 O15244 1/20 0.47
CACNA1F O60840 1/20 0.47
ADRB2 P07550 1/20 0.47
CHRM2 P08172 1/20 0.47
CHRM4 P08173 1/20 0.47
CHRM5 P08912 1/20 0.47
ADRA2A P08913 1/20 0.47
CYP2D6 P10635 1/20 0.47
CHRM1 P11229 1/20 0.47
ADRA2B P18089 1/20 0.47
ADRA2C P18825 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9535893 0.87 HTR1A (0.53) DRD2HTR2AHTR1AKCNH2HTR2C
SCHEMBL9537098 0.85 HTR2A (0.49) DRD2HTR2AHTR1AKCNH2HTR2C
SCHEMBL9536489 0.84 ADRA1A (0.48) DRD2HTR2AHTR1AHTR2CADRA1A
SCHEMBL10551226 0.77 DRD2 (0.52) DRD2HTR2AHTR1AKCNH2HTR2C
SCHEMBL10551137 0.77 DRD2 (0.52) DRD2HTR2AHTR1AKCNH2HTR2C
SCHEMBL9537863 0.76 SSTR5 (0.45) DRD2HTR2AHTR1AKCNH2HTR2C
SCHEMBL9537922 0.75 ALDH1A1 (0.38) DRD2HTR2AHTR1ATSHRKDM4E
SCHEMBL9537833 0.75 ALDH1A1 (0.39) DRD2HTR2AHTR1ATSHRDRD4
SCHEMBL9538362 0.74 ACHE (0.48) DRD2HTR2AHTR1AKCNH2HTR2C
SCHEMBL10549621 0.74 SLC6A9 (0.53) DRD2HTR2AHTR1AKCNH2HTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0151826-B1 4-[(Bicyclic heterocyclyl)-methyl and -hetero]-piperidines JANSSEN PHARMACEUTICA N.V. (BE) 1993-03-31 EP claimed