SCHEMBL959018

SCHEMBL959018

CC(=O)CNC(=O)OC(C)(C)C

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.50
MAOA P21397 1/20 0.47
MAOB P27338 1/20 0.47
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
GAA P10253 1/20 0.47
ALDH1A1 P00352 1/20 0.42
TSHR P16473 1/20 0.42
CA2 P00918 4/20 0.42
CA12 O43570 4/20 0.42
CA14 Q9ULX7 2/20 0.42
CA1 P00915 4/20 0.41
CA9 Q16790 2/20 0.41
EPHX1 P07099 1/20 0.41
CA7 P43166 2/20 0.40
KDM4E B2RXH2 1/20 0.38
LMNA P02545 1/20 0.38
APLNR P35414 1/20 0.38
CTSS P25774 2/20 0.38
CTSK P43235 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12201805 0.92 TDP1 (0.44) TDP1MAOAMAOBMEN1KMT2A
SCHEMBL3642785 0.92 MAOA (0.46) TDP1MAOAMAOBMEN1KMT2A
SCHEMBL27429142 0.86 TDP1 (0.50) TDP1MAOAMAOBMEN1KMT2A
SCHEMBL15931183 0.85 TDP1 (0.46) TDP1MAOAMAOBMEN1KMT2A
SCHEMBL21962098 0.84 MEN1 (0.50) TDP1MAOAMAOBMEN1KMT2A
SCHEMBL125503 0.84 TDP1 (0.52) TDP1MAOAMAOBMEN1KMT2A
SCHEMBL4714065 0.84 TDP1 (0.52) TDP1MAOAMAOBMEN1KMT2A
SCHEMBL6234096 0.83 TDP1 (0.49) TDP1MAOAMAOBMEN1KMT2A
SCHEMBL18618701 0.83 TDP1 (0.47) TDP1MAOAMAOBMEN1KMT2A
SCHEMBL3131272 0.83 TDP1 (0.47) TDP1MAOAMAOBMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 157 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114751867-A Feed additive capable of improving immunity and preparation method and application thereof 河南湾流生物科技有限公司 2022-07-15 CN claimed
CN-105018541-B (S) synthetic method of the hydroxy propyl carbamate of the tert-butyl group 2 上海合全药物研发有限公司 2018-03-27 CN claimed
CN-105018541-A Synthetic method of (S)-t-butyl-2-hydroxypropylcarbamate SHANGHAI SYNTHEALL PHARMACEUTICALS RES CO LTD 2015-11-04 CN claimed
EP-3941459-B1 QUINOLINE AND QUINAZOLINE COMPOUNDS AND METHODS OF USE THEREOF STINGRAY THERAPEUTICS INC (US) 2026-05-06 EP disclosed
WO-2026085629-A1 SUBSTITUTED HETEROCYCLIC COMPOUNDS, COMPOSITIONS COMPRISING THEM AND USES THEREOF Université de Montréal (CA) 2026-04-30 WO disclosed
US-20260015350-A1 AZAQUINAZOLINE PAN-KRAS INHIBITORS MIRATI THERAPEUTICS INC (US) 2026-01-15 US disclosed
US-12398120-B2 Substituted hydantoinamides as ADAMTS7 antagonists BAYER AKTIENGESELLSCHAFT (DE) 2025-08-26 US disclosed
EP-4058452-B1 HYDROPYRAZINO[1,2-B]ISOQUINOLINE COMPOUNDS FOR THE TREATMENT OF AUTOIMMUNE DISEASE HOFFMANN LA ROCHE (CH) 2025-07-09 EP disclosed
EP-4540255-A1 AZAQUINAZOLINE PAN-KRAS INHIBITORS Mirati Therapeutics, Inc. (US) 2025-04-23 EP disclosed
US-20250092016-A1 COMPOUNDS AND COMPOSITIONS FOR THE TREATMENT OF CORONAVIRAL RELATED DISEASES NOVARTIS AG (CH) 2025-03-20 US disclosed
US-20250074909-A1 AMINOTRIAZOLOPYRIDINES AS KINASE INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2025-03-06 US disclosed
US-20070099841-A1 Prodrugs of T3 and T4 with enhanced bioavailability NEW RIVER PHARMACEUTICALS INC. (US) 2007-05-03 US disclosed
EP-1771443-A1 QUINOLINE THIAZOLINONES WITH CDK1 ANTIPROLIFERATIVE ACTIVITY F.HOFFMANN-LA ROCHE AG (CH) 2007-04-11 EP disclosed
WO-2007020194-A1 PIPERIDINE AND PIPERAZINE DERIVATIVES AS P2X3 ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2007-02-22 WO disclosed
WO-2006104356-A1 DIPEPTIDYL PEPTIDASE-IV INHIBITING COMPOUNDS, METHODS OF PREPARING THE SAME, AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME AS AN ACTIVE AGENT LG LIFE SCIENCES, LTD. (KR) 2006-10-05 WO disclosed
WO-2006002828-A1 QUINOLINE THIAZOLINONES WITH CDK1 ANTIPROLIFERATIVE ACTIVITY F. HOFFMANN-LA ROCHE AG (CH) 2006-01-12 WO disclosed
US-20060004046-A1 Thiazolinone 3,4-disubstituted quinolines CHEN LI 2006-01-05 US disclosed
CN-1202096-C 2-aminothiazoline derivatives and their use as no-synthase inhibitors AVENTIS PHARMA SA (FR) 2005-05-18 CN disclosed
CN-1444572-A 2-aminothiazoline derivatives and their use as no-synthase inhibitors AVENTIS PHARMA SA (FR) 2003-09-24 CN disclosed
WO-1995033724-A1 PHENETHANOLAMINE DERIVATIVES AND THEIR USE AS ATYPICAL BETA-ADRENOCEPTOR AGONISTS GLAXO GROUP LIMITED (GB) 1995-12-14 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250092016-A1 COMPOUNDS AND COMPOSITIONS FOR THE TREATMENT OF CORONAVIRAL RELATED DISEASES ACE2, ACE, TMPRSS2 TDP1 3482/4885MAOA 353/4885MAOB 372/4885
US-20250074909-A1 AMINOTRIAZOLOPYRIDINES AS KINASE INHIBITORS RIPK1, RIPK3, RIPK4 TDP1 473/4885MAOA 4171/4885MAOB 3963/4885
US-12398120-B2 Substituted hydantoinamides as ADAMTS7 antagonists ADAMTS7, MMP7, ADAM17 TDP1 388/4885MAOA 1338/4885MAOB 1041/4885
US-20070099841-A1 Prodrugs of T3 and T4 with enhanced bioavailability THRA, THRB, SLC7A1 TDP1 723/4885MAOA 2604/4885MAOB 1940/4885
US-20060004046-A1 Thiazolinone 3,4-disubstituted quinolines CDK1, CDK17, CDK14 TDP1 787/4885MAOA 4524/4885MAOB 4378/4885
US-20260015350-A1 AZAQUINAZOLINE PAN-KRAS INHIBITORS KRAS, NRAS, HRAS TDP1 3609/4885MAOA 4857/4885MAOB 4796/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.