SCHEMBL9609560

SCHEMBL9609560

CC(C)(C)c1cnc2ccccn12

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SSTR4 P31391 1/20 0.48
NPSR1 Q6W5P4 2/20 0.46
FLT3 P36888 3/20 0.45
ADORA3 P0DMS8 1/20 0.43
GGPS1 O95749 1/20 0.42
FDPS P14324 1/20 0.42
DYRK1A Q13627 1/20 0.42
MIF P14174 1/20 0.41
NPC1 O15118 3/20 0.41
ALDH1A1 P00352 2/20 0.41
HPGD P15428 2/20 0.41
KDM4E B2RXH2 1/20 0.41
GLA P06280 1/20 0.41
GAA P10253 1/20 0.41
CASP1 P29466 1/20 0.41
CASP7 P55210 1/20 0.41
HSD17B10 Q99714 1/20 0.41
PKM P14618 1/20 0.41
PIK3CA P42336 1/20 0.40
RAB9A P51151 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27221248 0.85 SSTR4 (0.49) SSTR4NPSR1FLT3ADORA3GGPS1
SCHEMBL9537296 0.85 SSTR4 (0.46) SSTR4NPSR1FLT3ADORA3GGPS1
SCHEMBL24349591 0.84 SSTR4 (0.54) SSTR4NPSR1FLT3ADORA3GGPS1
SCHEMBL12463958 0.82 SSTR4 (0.44) SSTR4NPSR1FLT3ADORA3GGPS1
SCHEMBL24348662 0.80 SSTR4 (0.43) SSTR4NPSR1FLT3ADORA3GGPS1
SCHEMBL24348668 0.80 GGPS1 (0.46) SSTR4NPSR1FLT3ADORA3GGPS1
SCHEMBL20439080 0.80 SSTR4 (0.45) SSTR4NPSR1FLT3ADORA3GGPS1
SCHEMBL24348667 0.77 SSTR4 (0.44) SSTR4NPSR1FLT3ADORA3GGPS1
SCHEMBL29412812 0.77 SSTR4 (0.41) SSTR4NPSR1FLT3ADORA3GGPS1
SCHEMBL9911038 0.77 ADORA3 (0.47) SSTR4NPSR1FLT3ADORA3DYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 203 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12016896-B2 Dipeptidomimetics as inhibitors of human immunoproteasomes CORNELL UNIVERSITY (US) 2024-06-25 US disclosed
US-20240025898-A1 HPK1 ANTAGONISTS AND USES THEREOF SCHRÖDINGER, INC. 2024-01-25 US disclosed
US-20240025898-A1 HPK1 ANTAGONISTS AND USES THEREOF SCHRÖDINGER, INC. 2024-01-25 US disclosed
US-11820766-B2 Monoacylglycerol lipase modulators JANSSEN PHARMACEUTICA NV (BE) 2023-11-21 US disclosed
US-11820766-B2 Monoacylglycerol lipase modulators JANSSEN PHARMACEUTICA NV (BE) 2023-11-21 US disclosed
US-20230271939-A1 4-ETHYNYLPYRIDINE DERIVATIVES USEFUL AS GCN2 INHIBITORS IP2IPO INNOVATIONS LIMITED (GB) 2023-08-31 US disclosed
US-20230271939-A1 4-ETHYNYLPYRIDINE DERIVATIVES USEFUL AS GCN2 INHIBITORS IP2IPO INNOVATIONS LIMITED (GB) 2023-08-31 US disclosed
WO-2023158795-A1 INHIBITORS OF RNA HELICASE DHX9 AND USES THEREOF ACCENT THERAPEUTICS, INC. (US) 2023-08-24 WO disclosed
WO-2023154519-A1 INHIBITORS OF RNA HELICASE DHX9 AND USES THEREOF ACCENT THERAPEUTICS, INC. (US) 2023-08-17 WO disclosed
US-20230250082-A1 4-ETHYNYLPYRIDINE DERIVATIVES USEFUL AS GCN2 INHIBITORS IP2IPO INNOVATIONS LIMITED (GB) 2023-08-10 US disclosed
US-7932246-B2 Histone deacetylase inhibitors CHROMA THERAPEUTICS LTD. (GB) 2011-04-26 US disclosed
US-20110059961-A1 4-SUBSTITUTED PYRIDIN-3-YL-CARBOXAMIDE COMPOUNDS AND METHODS OF USE GENENTECH, INC. 2011-03-10 US disclosed
US-20110059961-A1 4-SUBSTITUTED PYRIDIN-3-YL-CARBOXAMIDE COMPOUNDS AND METHODS OF USE GENENTECH, INC. 2011-03-10 US disclosed
US-20100317678-A1 HYDROXAMATES AS INHIBITORS OF HISTONE DEACETYLASE CHROMA THERAPEUTICS LTD. (GB) 2010-12-16 US disclosed
US-20100190777-A1 COMPOUNDS AND METHODS FOR KINASE MODULATION, AND INDICATIONS THEREFOR PLEXXIKON INC. (US) 2010-07-29 US disclosed
US-20100152155-A1 Histone Deacetylase Inhibitors CHROMA THERAPEUTICS LTD. (GB) 2010-06-17 US disclosed
US-20090298924-A1 HYDROXAMIC ACID DERIVATIVES AS INHIBITORS OF HDAC ENZYMATIC ACTIVITY CHROMA THERAPEUTICS LTD (GB) 2009-12-03 US disclosed
US-20090298924-A1 HYDROXAMIC ACID DERIVATIVES AS INHIBITORS OF HDAC ENZYMATIC ACTIVITY CHROMA THERAPEUTICS LTD (GB) 2009-12-03 US disclosed
US-20090291978-A1 Enzyme Inhibitors CHROMA THERAPEUTICS LTD. (GB) 2009-11-26 US disclosed
US-20070191376-A1 Bicyclic heteroaryl compounds TAKEDA PHARMACEUTICALS U.S.A., INC. 2007-08-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (12 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230271939-A1 4-ETHYNYLPYRIDINE DERIVATIVES USEFUL AS GCN2 INHIBITORS EIF2AK4, GCN1, EIF5B SSTR4 3634/4885NPSR1 4053/4885FLT3 4318/4885
US-20100317678-A1 HYDROXAMATES AS INHIBITORS OF HISTONE DEACETYLASE H1-2, HDAC1, H1-0 SSTR4 3885/4885NPSR1 2488/4885FLT3 2698/4885
US-20230250082-A1 4-ETHYNYLPYRIDINE DERIVATIVES USEFUL AS GCN2 INHIBITORS EIF2AK4, GCN1, EIF5B SSTR4 3634/4885NPSR1 4053/4885FLT3 4318/4885
US-20070191376-A1 Bicyclic heteroaryl compounds CYP3A43, CYP11B2, CYP2F1 SSTR4 1933/4885NPSR1 726/4885FLT3 489/4885
US-20090298924-A1 HYDROXAMIC ACID DERIVATIVES AS INHIBITORS OF HDAC ENZYMATIC ACTIVITY HDAC1, HDAC3, HAT1 SSTR4 3089/4885NPSR1 745/4885FLT3 2166/4885
US-20240025898-A1 HPK1 ANTAGONISTS AND USES THEREOF PDXK, HIPK1, PCK1 SSTR4 3641/4885NPSR1 2913/4885FLT3 2057/4885
US-20100190777-A1 COMPOUNDS AND METHODS FOR KINASE MODULATION, AND INDICATIONS THEREFOR MAP3K20, MAP3K11, MAP3K10 SSTR4 3365/4885NPSR1 2686/4885FLT3 346/4885
US-20090291978-A1 Enzyme Inhibitors HAT1, NR2E1, NR2C2 SSTR4 3414/4885NPSR1 2152/4885FLT3 2174/4885
US-20110059961-A1 4-SUBSTITUTED PYRIDIN-3-YL-CARBOXAMIDE COMPOUNDS AND METHODS OF USE PIM1, PIM3, PIM2 SSTR4 3453/4885NPSR1 4623/4885FLT3 34/4885
US-11820766-B2 Monoacylglycerol lipase modulators MGLL, LPL, PNLIP SSTR4 2673/4885NPSR1 712/4885FLT3 2356/4885
US-12016896-B2 Dipeptidomimetics as inhibitors of human immunoproteasomes PREP, CTSC, DNPEP SSTR4 1198/4885NPSR1 565/4885FLT3 1047/4885
US-20100152155-A1 Histone Deacetylase Inhibitors HDAC1, HDAC2, HDAC11 SSTR4 4330/4885NPSR1 3160/4885FLT3 3620/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.