SCHEMBL9645653

SCHEMBL9645653

O=C1CCCN(c2cccc(COCc3ccccc3)c2)N1Cc1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
APP P05067 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.41
GRM5 P41594 2/20 0.39
CACNA2D1 P54289 1/20 0.39
AGXT P21549 1/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
TSHR P16473 1/20 0.37
PARP1 P09874 1/20 0.36
LMNA P02545 3/20 0.36
ALDH1A1 P00352 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
HPGD P15428 1/20 0.36
CYP2C19 P33261 1/20 0.36
ALOX5 P09917 2/20 0.36
GAA P10253 2/20 0.36
MAPT P10636 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9645284 0.84 L3MBTL1 (0.51) L3MBTL1NPC1RAB9AALOX5GAA
SCHEMBL9645861 0.81 GRM5 (0.40) APPL3MBTL1GRM5NPC1RAB9A
SCHEMBL9645378 0.72 ALOX5 (0.68) APPALOX5
SCHEMBL13097411 0.67 GRM5 (0.56) L3MBTL1GRM5CACNA2D1NPC1RAB9A
SCHEMBL6947156 0.67 CASP1 (0.53) L3MBTL1TSHRALDH1A1
SCHEMBL791963 0.66 ALDH1A1 (0.54) L3MBTL1CACNA2D1NPC1RAB9ATSHR
SCHEMBL7279696 0.65 PKM (0.63) L3MBTL1NPC1RAB9ATSHRLMNA
SCHEMBL10415710 0.65 ALDH1A1 (0.47) L3MBTL1TSHRLMNAALDH1A1CYP1A2
SCHEMBL10417568 0.65 MGLL (0.43) ALDH1A1CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL29007243 0.65 TSHR (0.79) APPL3MBTL1AGXTTSHRMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5086052-A Antiarthritic, antiallergens, antiinflammatory agents; also for asthma and psoriasis ABBOTT LABORATORIES (US) 1992-02-04 US disclosed
US-4970210-A ENZYME INHIBITORS ABBOTT LABORATORIES (US) 1990-11-13 US disclosed
EP-0299449-A2 Pyridazinone, triazinone and oxapyridazinone lipoxygenase inhibiting compounds ABBOTT LABORATORIES (US) 1989-01-18 EP disclosed