SCHEMBL9720347

SCHEMBL9720347

CCC(C)C(C(=O)[O-])C(C)(O)c1cnccn1.[Na+]

nearest known ligand 0.35

Known targets — ChEMBL curated mechanism

ABCC8ACEADORA1ADORA2AADORA2BADORA3ALDH5A1ALOX5ALOX5APATP4AATP4BBRAFCA1CA12CA2CA4CYSLTR1DHFRDPEP1EDNRAEDNRBESR2F10FDPSFGF1GABBR1GABBR2GABRA1GABRA2GABRA3GABRA4GABRA5GABRA6GABRB1GABRB2GABRB3GABRDGABREGABRG1GABRG2GABRG3GABRPGABRQGARTGNRHRGSC1HMGCRIMPDH1IMPDH2KCNJ11LY96NOD2NR3C1NS3NS4ANS5bP2RY1P2RY12P2RY2P2RY4P2RY6PBP2XPDE3APDE3BPDE4APDE4BPDE4CPDE4DPDK1PDK2PDK3PDK4PPARGPPATPTGIRPTGS1PTGS2RAF1RYR1RYR3SCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASERPINC1SLC12A1SLC12A3SYKTHRATHRBTLR3TLR4TLR9TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYMSVKORC1XDHblablaIMP-1blaOXA-33blaOXA-58blaT-3blaT-4blaT-5blaT-6dacAdacBdacCfolAfolPfolP1ftsIfusAgaggyrAgyrBmecAmrcAmrcBmrdApbp1apbp1bpbp2pbp2apbp2bpbp3pbp4pbpApbpBpbpCpbpFpolponBrplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpoArpoBrpoCrpoZrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of None. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
THRB known ✓ P10828 1/20 0.32
ABCC8 known ✓ Q09428 1/20 0.31
KCNJ11 known ✓ Q14654 1/20 0.31
CYP19A1 P11511 1/20 0.35
POLB P06746 1/20 0.34
KDM4E B2RXH2 3/20 0.33
RAB9A P51151 2/20 0.33
KMT2A Q03164 1/20 0.33
LONP1 P36776 3/20 0.32
HTT P42858 2/20 0.32
LMNA P02545 2/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
GAA P10253 1/20 0.32
NPC1 O15118 1/20 0.31
ABCC9 O60706 1/20 0.31
KCNJ8 Q15842 1/20 0.31
MLYCD O95822 1/20 0.30
ALDH1A1 P00352 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9720324 0.86 LMNA (0.39) CYP19A1POLBKDM4ERAB9AKMT2A
Ammonia Solution, Strong SCHEMBL9720328 0.85 LMNA (0.38) CYP19A1POLBKDM4ERAB9AKMT2A
SCHEMBL11068158 0.83 SMN1; SMN2 (0.37) CYP19A1POLBKDM4ERAB9AKMT2A
SCHEMBL9720326 0.78 CYP3A4 (0.42) CYP19A1RAB9AKMT2ALMNANPC1
SCHEMBL9720319 0.77 CYP19A1 (0.33) CYP19A1KMT2AHTTLMNASMN1; SMN2
SCHEMBL781412 0.71 CYP19A1 (0.43) CYP19A1POLBKDM4ERAB9ALONP1
SCHEMBL781413 0.71 CYP19A1 (0.43) CYP19A1POLBKDM4ERAB9ALONP1
SCHEMBL26833406 0.71 CYP19A1 (0.43) CYP19A1POLBKDM4ERAB9ALONP1
SCHEMBL9720300 0.66 RAB9A (0.34) KDM4ERAB9AKMT2ALONP1HTT
SCHEMBL10701851 0.64 KDM4E (0.41) CYP19A1POLBKDM4ERAB9AKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5148817-A Heterocyclic hydroxy-substituted carboxylic compound as flavor additive PHILIP MORRIS INCORPORATED (US) 1992-09-22 US claimed