SCHEMBL9724095

SCHEMBL9724095

COc1ccc(Sc2ccc(CNO)s2)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.40
POLB P06746 3/20 0.40
MMP2 P08253 3/20 0.40
MMP9 P14780 3/20 0.40
MMP12 P39900 3/20 0.40
KMT2A Q03164 2/20 0.40
MMP14 P50281 1/20 0.40
MEN1 O00255 1/20 0.40
PTGIR P43119 3/20 0.39
GAA P10253 3/20 0.37
KDM4E B2RXH2 2/20 0.37
MAPT P10636 2/20 0.37
HTT P42858 2/20 0.37
L3MBTL1 Q9Y468 2/20 0.37
MTNR1A P48039 1/20 0.35
MTNR1B P49286 1/20 0.35
CYP1A1 P04798 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP1B1 Q16678 1/20 0.35
ALDH1A1 P00352 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9724093 0.80 MEN1 (0.33) POLBKMT2AMEN1PTGIRMAPT
SCHEMBL9724109 0.80 THRB (0.39) TP53POLBMMP2KMT2AMEN1
SCHEMBL9724097 0.73 ALOX5 (0.41) MMP2MMP9MMP12PTGIR
SCHEMBL11521743 0.72 LTA4H (0.51) POLBKMT2AMEN1PTGIRKDM4E
SCHEMBL11398559 0.70 PKM (0.53) TP53POLBMMP2MMP9MMP12
SCHEMBL7593054 0.68 ALDH1A1 (0.43) PTGIRMAPTCYP1A1CYP1A2CYP1B1
SCHEMBL482369 0.67 CA1 (0.65) POLBKMT2AMEN1PTGIRGAA
SCHEMBL157282 0.66 ALDH1A1 (0.62) KMT2AMEN1GAAMAPTHTT
SCHEMBL9724126 0.66 KDM4E (0.47) POLBGAAKDM4EMAPTL3MBTL1
Hydrochloric Acid SCHEMBL11848856 0.65 CA1 (0.61) POLBKMT2AMEN1PTGIRGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5158971-A Antiallergens, antiinflammatory agents LILLY INDUSTRIES LIMITED (GB) 1992-10-27 US disclosed
EP-0459748-A2 Thien-2-yl methylurea derivatives as leukotriene inhibitors LILLY INDUSTRIES LIMITED (GB) 1991-12-04 EP disclosed