SCHEMBL9727633

SCHEMBL9727633

COC1Oc2cc(CCCO)c(OCc3ccccc3)cc2C1(C)C

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 1/20 0.38
EPHX2 P34913 1/20 0.38
MTNR1A P48039 3/20 0.37
MTNR1B P49286 2/20 0.37
PTGER1 P34995 3/20 0.37
PTGER4 P35408 3/20 0.37
PTGER3 P43115 3/20 0.37
PTGER2 P43116 3/20 0.37
AKR1B1 P15121 1/20 0.36
RRM1 P23921 1/20 0.35
HTR6 P50406 1/20 0.35
ALDH1A1 P00352 1/20 0.34
DUSP3 P51452 1/20 0.34
ABCB1 P08183 1/20 0.34
HTR1A P08908 1/20 0.34
DRD2 P14416 1/20 0.34
NR3C1 P04150 1/20 0.34
CYP4F2 P78329 1/20 0.33
CYP4A11 Q02928 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9727700 0.90 MTNR1A (0.35) MTNR1AMTNR1BPTGER1PTGER4PTGER3
SCHEMBL9727653 0.89 ABCB1 (0.38) MTNR1AMTNR1BPTGER1PTGER4PTGER3
SCHEMBL9727762 0.82 NR3C1 (0.38) AKR1B1ALDH1A1ABCB1HTR1ADRD2
SCHEMBL9727331 0.77 MTNR1A (0.37) MTNR1AMTNR1BPTGER1PTGER4PTGER3
SCHEMBL14552343 0.74 MAOB (0.52) LTA4HEPHX2PTGER1PTGER4PTGER3
SCHEMBL9727686 0.71 NR3C1 (0.38) PTGER1PTGER4PTGER3PTGER2AKR1B1
SCHEMBL9727488 0.71 ABCB1 (0.43) LTA4HEPHX2MTNR1AMTNR1BABCB1
SCHEMBL14435033 0.69 HTR6 (0.43) LTA4HEPHX2PTGER1PTGER4PTGER3
SCHEMBL10460139 0.69 LTA4H (0.43) LTA4HEPHX2MTNR1AMTNR1BPTGER1
SCHEMBL31561714 0.67 HTR1A (0.69) LTA4HEPHX2PTGER1PTGER4PTGER3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5091533-A Treating allergies, cardiovascular disorders, inflammation MERCK FROSST CANADA, INC. (CA) 1992-02-25 US disclosed
EP-0447189-A1 5-Hydroxy-2,3-dihydrobenzofuran analogs as leukotriene biosynthesis inhibitors MERCK FROSST CANADA INC. (CA) 1991-09-18 EP disclosed