SCHEMBL9727686

SCHEMBL9727686

C=CCc1cc2c(cc1OCc1ccccc1)C(C)(C)C(CCO)O2

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR3C1 P04150 1/20 0.38
AKR1B1 P15121 1/20 0.35
ALDH1A1 P00352 3/20 0.35
MAPT P10636 2/20 0.35
GAA P10253 1/20 0.35
HPGD P15428 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
PTPN1 P18031 1/20 0.34
SIRT1 Q96EB6 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
KDM4E B2RXH2 2/20 0.32
PTGER1 P34995 1/20 0.32
PTGER4 P35408 1/20 0.32
PTGER3 P43115 1/20 0.32
PTGER2 P43116 1/20 0.32
POLB P06746 1/20 0.32
HIF1A Q16665 1/20 0.32
USP28 Q96RU2 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9727307 0.86 L3MBTL1 (0.36) NR3C1AKR1B1ALDH1A1MAPTGAA
SCHEMBL9727725 0.84 AKR1B1 (0.32) NR3C1AKR1B1ALDH1A1MAPTGAA
SCHEMBL9727762 0.82 NR3C1 (0.38) NR3C1AKR1B1ALDH1A1MAPTGAA
SCHEMBL9727633 0.71 LTA4H (0.38) NR3C1AKR1B1ALDH1A1PTGER1PTGER4
SCHEMBL9727777 0.71 AKR1B1 (0.35) AKR1B1ALDH1A1GAAKMT2AKDM4E
SCHEMBL14552348 0.71 MAOB (0.54) ALDH1A1MAPTGAAHPGDTDP1
SCHEMBL9727331 0.67 MTNR1A (0.37) AKR1B1PTGER1PTGER4PTGER3PTGER2
SCHEMBL9727671 0.67 MAOB (0.46) HIF1A
SCHEMBL9727700 0.65 MTNR1A (0.35) AKR1B1MAPTTDP1L3MBTL1PTGER1
SCHEMBL9727653 0.65 ABCB1 (0.38) PTGER1PTGER4PTGER3PTGER2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5091533-A Treating allergies, cardiovascular disorders, inflammation MERCK FROSST CANADA, INC. (CA) 1992-02-25 US disclosed
EP-0447189-A1 5-Hydroxy-2,3-dihydrobenzofuran analogs as leukotriene biosynthesis inhibitors MERCK FROSST CANADA INC. (CA) 1991-09-18 EP disclosed