SCHEMBL9727700

SCHEMBL9727700

COC1Oc2cc(CCCBr)c(OCc3ccccc3)cc2C1(C)C

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 3/20 0.35
MTNR1B P49286 2/20 0.35
PTGER1 P34995 2/20 0.35
PTGER4 P35408 2/20 0.35
PTGER3 P43115 2/20 0.35
PTGER2 P43116 2/20 0.35
AKR1B1 P15121 1/20 0.34
ABCB1 P08183 4/20 0.34
HTR1A P08908 2/20 0.34
DRD2 P14416 2/20 0.34
L3MBTL1 Q9Y468 2/20 0.32
ABCG2 Q9UNQ0 1/20 0.32
MAPT P10636 1/20 0.32
MAPK1 P28482 1/20 0.32
TDP1 Q9NUW8 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9727633 0.90 LTA4H (0.38) MTNR1AMTNR1BPTGER1PTGER4PTGER3
SCHEMBL9727653 0.89 ABCB1 (0.38) MTNR1AMTNR1BPTGER1PTGER4PTGER3
SCHEMBL9727762 0.82 NR3C1 (0.38) AKR1B1ABCB1HTR1ADRD2L3MBTL1
SCHEMBL9727331 0.75 MTNR1A (0.37) MTNR1AMTNR1BPTGER1PTGER4PTGER3
SCHEMBL9727567 0.69 CYP3A4 (0.37) PTGER1PTGER4PTGER3PTGER2HTR1A
SCHEMBL4951651 0.67 ALOX5 (0.49) PTGER1PTGER4PTGER3PTGER2ABCB1
SCHEMBL9727777 0.67 AKR1B1 (0.35) AKR1B1ABCB1HTR1ADRD2ABCG2
SCHEMBL9727620 0.65 CCR5 (0.38) PTGER1PTGER4PTGER3PTGER2
SCHEMBL21363672 0.64 MAOB (0.52) MTNR1APTGER1PTGER4PTGER3PTGER2
SCHEMBL21363757 0.62 MAOB (0.50) MTNR1APTGER1PTGER4PTGER3PTGER2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5091533-A Treating allergies, cardiovascular disorders, inflammation MERCK FROSST CANADA, INC. (CA) 1992-02-25 US disclosed
EP-0447189-A1 5-Hydroxy-2,3-dihydrobenzofuran analogs as leukotriene biosynthesis inhibitors MERCK FROSST CANADA INC. (CA) 1991-09-18 EP disclosed