SCHEMBL9727777

SCHEMBL9727777

CCCc1cc2c(cc1OCc1ccccc1)C(C)(C)C(CCc1ccc(SC)cc1)O2

nearest known ligand 0.67

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 1/20 0.35
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
POLB P06746 1/20 0.32
KMT2A Q03164 1/20 0.32
ABCB1 P08183 2/20 0.32
HTR1A P08908 1/20 0.32
DRD2 P14416 1/20 0.32
GCK P35557 2/20 0.32
SIRT2 Q8IXJ6 1/20 0.31
ABCG2 Q9UNQ0 1/20 0.31
LMNA P02545 1/20 0.31
GAA P10253 1/20 0.31
FFAR1 O14842 1/20 0.31
FFAR4 Q5NUL3 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9727725 0.88 AKR1B1 (0.32) AKR1B1ALDH1A1ABCB1HTR1ADRD2
SCHEMBL9727660 0.80 CGAS (0.31) LMNA
SCHEMBL9727464 0.78 KDM4E (0.36) AKR1B1KDM4EALDH1A1KMT2ALMNA
SCHEMBL9727686 0.71 NR3C1 (0.38) AKR1B1KDM4EALDH1A1POLBKMT2A
SCHEMBL9727307 0.67 L3MBTL1 (0.36) AKR1B1KDM4EALDH1A1POLBKMT2A
SCHEMBL9727331 0.67 MTNR1A (0.37) AKR1B1ABCB1HTR1ADRD2
SCHEMBL9727633 0.67 LTA4H (0.38) AKR1B1ALDH1A1ABCB1HTR1ADRD2
SCHEMBL9727700 0.67 MTNR1A (0.35) AKR1B1ABCB1HTR1ADRD2ABCG2
SCHEMBL21363788 0.67 MAOB (0.55) ALDH1A1KMT2AHTR1ADRD2GAA
SCHEMBL9727653 0.66 ABCB1 (0.38) ABCB1HTR1ADRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5091533-A Treating allergies, cardiovascular disorders, inflammation MERCK FROSST CANADA, INC. (CA) 1992-02-25 US disclosed
EP-0447189-A1 5-Hydroxy-2,3-dihydrobenzofuran analogs as leukotriene biosynthesis inhibitors MERCK FROSST CANADA INC. (CA) 1991-09-18 EP disclosed