SCHEMBL9737119

SCHEMBL9737119

CC(=O)Nc1ccc2c(c1)C(n1ccccc1=O)C(O)C(C)(C)C2

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 2/20 0.40
CYP1A2 P05177 1/20 0.40
ADRA2A P08913 1/20 0.40
SLC6A2 P23975 1/20 0.40
HTR2C P28335 1/20 0.40
SLC6A4 P31645 1/20 0.40
HTR2B P41595 1/20 0.40
ALDH1A1 P00352 4/20 0.39
KDM4E B2RXH2 2/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
SIGMAR1 Q99720 1/20 0.39
NPC1 O15118 2/20 0.38
RAB9A P51151 2/20 0.38
MAPT P10636 3/20 0.37
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
PDK2 Q15119 2/20 0.37
KDM4A O75164 1/20 0.37
POLB P06746 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9732909 0.85 OPRD1 (0.35) ALDH1A1KDM4EL3MBTL1MAPT
SCHEMBL9735080 0.81 TSHR (0.42) HTR2CHTR2BALDH1A1KDM4ENPC1
SCHEMBL9733607 0.81 DRD1 (0.35) ALDH1A1KDM4ESIGMAR1MAPTSMN1; SMN2
SCHEMBL9733666 0.81 ALDH1A1 (0.38) SLC6A2SLC6A4ALDH1A1KDM4EL3MBTL1
SCHEMBL8088757 0.80 ABCC9 (0.41) MAOACYP1A2MAPTMEN1KMT2A
SCHEMBL9733350 0.78 HIF1A (0.41) ALDH1A1MAPTSMN1; SMN2HTR2A
SCHEMBL9734096 0.78 ABCC9 (0.41) CYP1A2
SCHEMBL9735453 0.77 TRPV1 (0.36) MAOACYP1A2ADRA2ASLC6A2HTR2C
SCHEMBL9596387 0.70 RAB9A (0.46) CYP1A2ALDH1A1KDM4EL3MBTL1NPC1
SCHEMBL8085317 0.70 MAOA (0.36) MAOACYP1A2ALDH1A1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5132307-A TETRALIN COMPOUNDS MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1992-07-21 US disclosed
EP-0368160-A1 Tetralin derivatives MERCK PATENT GmbH (DE) 1990-05-16 EP disclosed