SCHEMBL9836563

SCHEMBL9836563

c1ccc2c(c1)Cc1cccnc1C(NCCN1CCCC1)O2

nearest known ligand 0.36

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ADRA2C P18825 7/20 0.36
ADRA2A P08913 6/20 0.36
ADRA2B P18089 6/20 0.36
HRH3 Q9Y5N1 1/20 0.36
ALOX15 P16050 1/20 0.35
TSHR P16473 1/20 0.35
CXCR4 P61073 1/20 0.35
LTA4H P09960 3/20 0.34
DPP7 Q9UHL4 1/20 0.34
CHRM2 P08172 1/20 0.34
CHRM4 P08173 1/20 0.34
CHRM5 P08912 1/20 0.34
CHRM1 P11229 1/20 0.34
CHRM3 P20309 1/20 0.34
SIGMAR1 Q99720 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9836619 0.91 CXCR4 (0.42) TSHRCXCR4LTA4HCHRM2CHRM4
SCHEMBL9836638 0.79 CYP2C19 (0.41) ADRA2CADRA2AADRA2BTSHRCHRM2
SCHEMBL9837035 0.79 OPRL1 (0.42) CXCR4LTA4H
SCHEMBL9835190 0.77 HTR1A (0.35) ADRA2CHRH3ALOX15LTA4HCHRM2
SCHEMBL9834580 0.76 HRH1 (0.36) ALOX15TSHRCXCR4CHRM2CHRM4
SCHEMBL9835645 0.76 ALDH1A1 (0.37) ADRA2CHRH3ALOX15TSHRLTA4H
SCHEMBL9836246 0.72 MTNR1A (0.40) TSHR
SCHEMBL9834815 0.70 CHRM2 (0.42) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL9835161 0.68 HRH3 (0.38) ADRA2CADRA2AADRA2BHRH3ALOX15
SCHEMBL9837005 0.68 MAOA (0.41)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0129879-B1 A [1] benzepino(3,4-b)pyridine derivative KYOWA HAKKO KOGYO CO., LTD. (JP) 1991-09-11 EP claimed
US-4547496-A Antiulcer [1] benzepino[3,4-b]pyridine and compositions KYOWA HAKKO KOGYO CO., LTD. (JP) 1985-10-15 US claimed