SCHEMBL9837035

SCHEMBL9837035

c1ccc2c(c1)Cc1cccnc1C(NCCCNC1CCCCC1)O2

nearest known ligand 0.42

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
OPRL1 P41146 3/20 0.42
CXCR4 P61073 9/20 0.41
CYP2D6 P10635 2/20 0.41
CYP3A4 P08684 1/20 0.41
GRIN1 Q05586 2/20 0.40
GRIN2B Q13224 2/20 0.40
LTA4H P09960 2/20 0.39
HTR1A P08908 2/20 0.38
HTR1D P28221 2/20 0.38
CXCL12 P48061 1/20 0.38
LMNA P02545 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9835645 0.79 ALDH1A1 (0.37) CYP2D6LTA4HHTR1AHTR1D
SCHEMBL9836563 0.79 ADRA2C (0.36) CXCR4LTA4H
SCHEMBL9836638 0.78 CYP2C19 (0.41) CYP2D6HTR1AHTR1DLMNA
SCHEMBL9835190 0.76 HTR1A (0.35) CYP2D6LTA4HHTR1AHTR1D
SCHEMBL9834580 0.76 HRH1 (0.36) CXCR4CYP3A4HTR1AHTR1D
SCHEMBL9836619 0.75 CXCR4 (0.42) CXCR4CYP2D6CYP3A4LTA4HLMNA
SCHEMBL9836246 0.71 MTNR1A (0.40) HTR1AHTR1DLMNA
SCHEMBL9835877 0.69 GRIN1 (0.42) OPRL1CXCR4CYP2D6CYP3A4GRIN1
SCHEMBL21784360 0.68 HDAC1 (0.51) OPRL1CXCR4CYP2D6CYP3A4GRIN1
SCHEMBL9837005 0.67 MAOA (0.41) OPRL1HTR1AHTR1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0129879-B1 A [1] benzepino(3,4-b)pyridine derivative KYOWA HAKKO KOGYO CO., LTD. (JP) 1991-09-11 EP claimed
EP-0129879-B1 A [1] benzepino(3,4-b)pyridine derivative KYOWA HAKKO KOGYO CO., LTD. (JP) 1991-09-11 EP disclosed