SCHEMBL986292

SCHEMBL986292

CC(=O)OC1CC(C)(C)N(OC(=O)CC(O)(CC(=O)O)C(=O)O)C(C)(C)C1

nearest known ligand 0.49

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.49
KMT2A Q03164 2/20 0.49
MEN1 O00255 1/20 0.45
GAA P10253 1/20 0.45
ALDH1A1 P00352 3/20 0.44
ESR1 P03372 1/20 0.44
HSD17B10 Q99714 1/20 0.44
KDM4E B2RXH2 1/20 0.34
LMNA P02545 1/20 0.34
MAPT P10636 1/20 0.34
ALOX15 P16050 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1232469 0.96 KMT2A (0.52) TSHRKMT2AMEN1GAAALDH1A1
Citric Acid SCHEMBL3802141 0.87 TSHR (0.45) TSHRKMT2AMEN1GAAALDH1A1
Citric Acid SCHEMBL3802147 0.87 TSHR (0.45) TSHRKMT2AMEN1GAAALDH1A1
Citric Acid SCHEMBL3801878 0.86 TSHR (0.44) TSHRKMT2AMEN1GAAALDH1A1
SCHEMBL1232593 0.86 KMT2A (0.49) TSHRKMT2AMEN1GAAALDH1A1
SCHEMBL7038092 0.84 ALDH1A1 (0.42) TSHRKMT2AALDH1A1KDM4ELMNA
Citric Acid SCHEMBL988186 0.84 ALDH1A1 (0.42) TSHRKMT2AMEN1GAAALDH1A1
Citric Acid SCHEMBL988184 0.84 ALDH1A1 (0.42) TSHRKMT2AMEN1GAAALDH1A1
Citric Acid SCHEMBL1232464 0.84 ALDH1A1 (0.42) TSHRKMT2AMEN1GAAALDH1A1
Citric Acid SCHEMBL985126 0.84 ALDH1A1 (0.42) TSHRKMT2AMEN1GAAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 64 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2464739-B1 METHODS IN CELL CULTURES, AND RELATED INVENTIONS, EMPLOYING CERTAIN ADDITIVES BASF SE (DE) 2016-01-13 EP claimed
US-8859235-B2 Methods in cell cultures, and related inventions, employing certain additives BASF SE (DE) 2014-10-14 US claimed
EP-1680541-B1 STABILIZED BODY CARE PRODUCTS, HOUSEHOLD PRODUCTS, TEXTILES AND FABRICS BASF SE (DE) 2012-12-19 EP claimed
US-20120164162-A1 METHODS IN CELL CULTURES, AND RELATED INVENTIONS, EMPLOYING CERTAIN ADDITIVES BASF SE (DE) 2012-06-28 US claimed
EP-2464739-A2 METHODS IN CELL CULTURES, AND RELATED INVENTIONS, EMPLOYING CERTAIN ADDITIVES BASF SE (DE) 2012-06-20 EP claimed
WO-2011018472-A2 METHODS IN CELL CULTURES, AND RELATED INVENTIONS, EMPLOYING CERTAIN ADDITIVES BASF SE (DE) 2011-02-17 WO claimed
US-7862746-B2 Stabilization of natural composites BASF SE. (DE) 2011-01-04 US claimed
EP-1499286-B1 STABILIZED BODY CARE PRODUCTS AND HOUSEHOLD PRODUCTS BASF SE (DE) 2010-04-07 EP claimed
US-20070079446-A1 Stabilized body care products, household products, textiles and fabrics CIBA SPECIALTY CHEMICALS CORP. 2007-04-12 US claimed
WO-2006087269-A1 STABILIZATION OF NATURAL COMPOSITES CIBA SPECIALTY CHEMICALS HOLDING INC. (CH) 2006-08-24 WO claimed
US-20060183821-A1 Stabilization of natural composites CIBA CORPORATION 2006-08-17 US claimed
EP-1680541-A2 STABILIZED BODY CARE PRODUCTS, HOUSEHOLD PRODUCTS, TEXTILES AND FABRICS Ciba SC Holding AG (CH) 2006-07-19 EP claimed
US-20050220727-A1 Stabilized body care products, household products, textiles and fabrics CIBA CORPORATION 2005-10-06 US claimed
WO-2005042828-A2 STABILIZED BODY CARE PRODUCTS, HOUSEHOLD PRODUCTS, TEXTILES AND FABRICS CIBA SPECIALTY CHEMICALS HOLDING INC. (CH) 2005-05-12 WO claimed
EP-1499286-A1 STABILIZED BODY CARE PRODUCTS, HOUSEHOLD PRODUCTS, TEXTILES AND FABRICS Ciba SC Holding AG (CH) 2005-01-26 EP claimed
WO-2003103622-A1 STABILIZED BODY CARE PRODUCTS, HOUSEHOLD PRODUCTS, TEXTILES AND FABRICS CIBA SPECIALTY CHEMICALS HOLDING INC. (CH) 2003-12-18 WO claimed
US-6500303-B1 DERIVATIVES OF 1-OXYL-2,2,6,6-TETRAMETHYL-PIPERIDIN-4-OL; PROTECTION FROM ULTRAVIOLET, FLUORESCENT AND SUN LIGHT EXPOSURE CIBA SPECIALTY CHEMICALS CORPORATION 2002-12-31 US claimed
US-20020124980-A1 Inhibition of pulp and paper yellowing using nitroxides, hydroxylamines and other coadditives SELTZER RAYMOND R (US) 2002-09-12 US claimed
US-6254724-B1 STABILIZING AMOUNT OF A HINDERED AMINE COMPOUND SELECTED DERIVATIVES OF 1-OXYL-2,2,6,6-TETRAMETHYL-PIPERIDIN-4-OL OR WHICH ARE THEIR HYDROXYLAMINE SALTS CIBA SPECIALTY CHEMICALS CORPORATION 2001-07-03 US claimed
US-10098849-B2 Anti-radical agents BASF SE (DE) 2018-10-16 US disclosed
US-9358195-B2 Stabilized body care products, household products, textiles and fabrics BASF SE (DE) 2016-06-07 US disclosed
EP-2464739-B1 METHODS IN CELL CULTURES, AND RELATED INVENTIONS, EMPLOYING CERTAIN ADDITIVES BASF SE (DE) 2016-01-13 EP disclosed
EP-2699727-B1 METHOD OF DYEING POLYESTER HUNTSMAN ADV MAT SWITZERLAND (CH) 2014-11-19 EP disclosed
US-8859235-B2 Methods in cell cultures, and related inventions, employing certain additives BASF SE (DE) 2014-10-14 US disclosed
EP-2699727-A1 METHOD OF DYEING POLYESTER Huntsman Advanced Materials (Switzerland) GmbH (CH) 2014-02-26 EP disclosed
US-20140041134-A1 Method of Dyeing Polyester HUNTSMAN INTERNATIONAL LLC (US) 2014-02-13 US disclosed
EP-1896550-B1 STABILIZED ELECTROCHROMIC MEDIA BASF SE (DE) 2013-08-14 EP disclosed
US-20120328541-A1 Anti-radical agents BASCHONG WERNER (CH) 2012-12-27 US disclosed
EP-1680541-B1 STABILIZED BODY CARE PRODUCTS, HOUSEHOLD PRODUCTS, TEXTILES AND FABRICS BASF SE (DE) 2012-12-19 EP disclosed
WO-2012143167-A1 METHOD OF DYEING POLYESTER HUNTSMAN ADVANCED MATERIALS (SWITZERLAND) GMBH (CH) 2012-10-26 WO disclosed
US-20120164162-A1 METHODS IN CELL CULTURES, AND RELATED INVENTIONS, EMPLOYING CERTAIN ADDITIVES BASF SE (DE) 2012-06-28 US disclosed
EP-2464739-A2 METHODS IN CELL CULTURES, AND RELATED INVENTIONS, EMPLOYING CERTAIN ADDITIVES BASF SE (DE) 2012-06-20 EP disclosed
WO-2011018472-A2 METHODS IN CELL CULTURES, AND RELATED INVENTIONS, EMPLOYING CERTAIN ADDITIVES BASF SE (DE) 2011-02-17 WO disclosed
US-7862746-B2 Stabilization of natural composites BASF SE. (DE) 2011-01-04 US disclosed
US-7718096-B2 Stabilized electrochromic media CIBA SPECIALTY CHEMICALS CORPORATION (US) 2010-05-18 US disclosed
EP-1499286-B1 STABILIZED BODY CARE PRODUCTS AND HOUSEHOLD PRODUCTS BASF SE (DE) 2010-04-07 EP disclosed
US-7678381-B2 Stabilized body care products, household products, textiles and fabrics CIBA SPECIALTY CHEMICALS CORPORATION (US) 2010-03-16 US disclosed
US-20090258041-A1 Protection of Oxidizable Agents CIBA CORP. 2009-10-15 US disclosed
US-20080305055-A1 Anti-Radical Agents CIBA CORPORATION 2008-12-11 US disclosed
EP-1896550-A1 STABILIZED ELECTROCHROMIC MEDIA Ciba Specialty Chemicals Holding Inc. (CH) 2008-03-12 EP disclosed
US-20070079446-A1 Stabilized body care products, household products, textiles and fabrics CIBA SPECIALTY CHEMICALS CORP. 2007-04-12 US disclosed
WO-2007003508-A1 STABILIZED ELECTROCHROMIC MEDIA CIBA SPECIALTY CHEMICALS HOLDING INC. (CH) 2007-01-11 WO disclosed
US-20070002423-A1 Stabilized electrochromic media CIBA SPECIALTY CHEMICALS CORP. 2007-01-04 US disclosed
WO-2006087269-A1 STABILIZATION OF NATURAL COMPOSITES CIBA SPECIALTY CHEMICALS HOLDING INC. (CH) 2006-08-24 WO disclosed
US-20060183821-A1 Stabilization of natural composites CIBA CORPORATION 2006-08-17 US disclosed
EP-1680541-A2 STABILIZED BODY CARE PRODUCTS, HOUSEHOLD PRODUCTS, TEXTILES AND FABRICS Ciba SC Holding AG (CH) 2006-07-19 EP disclosed
EP-1230276-B1 PHOTOINITIATOR FORMULATIONS CIBA SC HOLDING AG (CH) 2005-12-14 EP disclosed
US-20050220727-A1 Stabilized body care products, household products, textiles and fabrics CIBA CORPORATION 2005-10-06 US disclosed
WO-2005042828-A2 STABILIZED BODY CARE PRODUCTS, HOUSEHOLD PRODUCTS, TEXTILES AND FABRICS CIBA SPECIALTY CHEMICALS HOLDING INC. (CH) 2005-05-12 WO disclosed
EP-1499286-A1 STABILIZED BODY CARE PRODUCTS, HOUSEHOLD PRODUCTS, TEXTILES AND FABRICS Ciba SC Holding AG (CH) 2005-01-26 EP disclosed
US-6803392-B1 AQUEOUS, STORAGE-STABLE, NON- SEDIMENTING SUSPENSIONS COMPRISING AT LEAST ONE MONO- OR BIS-ACYLPHOSPHINE OXIDE CIBA SPECIALTY CHEMICALS CORPORATION 2004-10-12 US disclosed
WO-2003103622-A1 STABILIZED BODY CARE PRODUCTS, HOUSEHOLD PRODUCTS, TEXTILES AND FABRICS CIBA SPECIALTY CHEMICALS HOLDING INC. (CH) 2003-12-18 WO disclosed
US-6630002-B2 Penetration, photostability and heat resistance with low solvent or solvent-free wood stains; dye stabilizer is a hydroxylamine or salt, preferably a 1-hydroxypiperidine CIBA SPECIALTY CHEMICALS CORPORATION 2003-10-07 US disclosed
EP-1280864-A1 PROCESS FOR THE STAINING OF WOOD WITH AQUEOUS WOOD STAINS Ciba SC Holding AG (CH) 2003-02-05 EP disclosed
US-6500303-B1 DERIVATIVES OF 1-OXYL-2,2,6,6-TETRAMETHYL-PIPERIDIN-4-OL; PROTECTION FROM ULTRAVIOLET, FLUORESCENT AND SUN LIGHT EXPOSURE CIBA SPECIALTY CHEMICALS CORPORATION 2002-12-31 US disclosed
US-20020124980-A1 Inhibition of pulp and paper yellowing using nitroxides, hydroxylamines and other coadditives SELTZER RAYMOND R (US) 2002-09-12 US disclosed
US-6447644-B1 PULP OR PAPER THAT STILL CONTAINS LIGNIN, AND A STERICALLY HINDERED AMINE, FOR EXAMPLE DERIVATIVES OF 1-OXYL-2,2,6,6-TETRAMETHYL-PIPERIDIN-4-OL CIBA SPECIALTY CHEMICALS CORPORATION 2002-09-10 US disclosed
EP-1230276-A1 PHOTOINITIATOR FORMULATIONS Ciba SC Holding AG (CH) 2002-08-14 EP disclosed
US-20020000011-A1 Process for the staining of wood with aqueous wood stains CIBA SPECIALTY CHEMICALSC CORP. 2002-01-03 US disclosed
WO-2001085857-A1 PROCESS FOR THE STAINING OF WOOD WITH AQUEOUS WOOD STAINS CIBA SPECIALTY CHEMICALS HOLDING INC. (CH) 2001-11-15 WO disclosed
US-6254724-B1 STABILIZING AMOUNT OF A HINDERED AMINE COMPOUND SELECTED DERIVATIVES OF 1-OXYL-2,2,6,6-TETRAMETHYL-PIPERIDIN-4-OL OR WHICH ARE THEIR HYDROXYLAMINE SALTS CIBA SPECIALTY CHEMICALS CORPORATION 2001-07-03 US disclosed
WO-2001029093-A1 PHOTOINITIATOR FORMULATIONS CIBA SPECIALTY CHEMICALS HOLDING INC. (CH) 2001-04-26 WO disclosed
EP-1000032-A1 INHIBITION OF PULP AND PAPER YELLOWING USING NITROXIDES AND OTHER COADDITIVES Ciba SC Holding AG (CH) 2000-05-17 EP disclosed
WO-1999005108-A1 INHIBITION OF PULP AND PAPER YELLOWING USING NITROXIDES AND OTHER COADDITIVES CIBA SPECIALTY CHEMICALS HOLDING INC. (CH) 1999-02-04 WO disclosed
WO-1999005108-A1 INHIBITION OF PULP AND PAPER YELLOWING USING NITROXIDES AND OTHER COADDITIVES CIBA SPECIALTY CHEMICALS HOLDING INC. (CH) 1999-02-04 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070079446-A1 Stabilized body care products, household products, textiles and fabrics CUTA, NISCH, DSC1 TSHR 1658/4885KMT2A 1072/4885MEN1 2500/4885
US-20120328541-A1 Anti-radical agents NOS3, GSTO1, TXN2 TSHR 3772/4885KMT2A 3587/4885MEN1 3889/4885
US-20050220727-A1 Stabilized body care products, household products, textiles and fabrics CUTA, DHRS9, DSC1 TSHR 1597/4885KMT2A 789/4885MEN1 2460/4885
US-20080305055-A1 Anti-Radical Agents NOS3, GSTO1, PTGS1 TSHR 3980/4885KMT2A 3828/4885MEN1 3539/4885
US-10098849-B2 Anti-radical agents NOS3, GSTO1, TXN2 TSHR 3772/4885KMT2A 3587/4885MEN1 3889/4885
US-20120164162-A1 METHODS IN CELL CULTURES, AND RELATED INVENTIONS, EMPLOYING CERTAIN ADDITIVES BBOX1, NEFM, NQO1 TSHR 4798/4885KMT2A 958/4885MEN1 3694/4885
US-20090258041-A1 Protection of Oxidizable Agents LPO, TYR, HAO2 TSHR 1453/4885KMT2A 3600/4885MEN1 4790/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.