SCHEMBL10475

SCHEMBL10475

CC1(C)OB(c2ccc3[nH]ncc3c2)OC1(C)C

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS1 P29475 4/20 0.45
ROCK2 O75116 4/20 0.45
MAPT P10636 2/20 0.45
ROCK1 Q13464 2/20 0.45
METAP2 P50579 1/20 0.45
CSNK2A1 P68400 1/20 0.45
KDM4E B2RXH2 1/20 0.45
MEN1 O00255 1/20 0.45
ALDH1A1 P00352 1/20 0.45
GAA P10253 1/20 0.45
HPGD P15428 1/20 0.45
RAB9A P51151 1/20 0.45
KMT2A Q03164 1/20 0.45
HIF1A Q16665 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
POLB P06746 1/20 0.43
MAOB P27338 1/20 0.43
GSK3B P49841 3/20 0.41
CLK1 P49759 2/20 0.41
DYRK3 O43781 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1318307 0.88 MAPT (0.45) NOS1MAPTMETAP2KDM4EMEN1
SCHEMBL29741038 0.88 MAPT (0.45) NOS1MAPTMETAP2KDM4EMEN1
SCHEMBL25234632 0.80 PRMT5 (0.47) ALDH1A1TDP1GSK3BLPLLIPG
SCHEMBL30399620 0.80 PRMT5 (0.47) ALDH1A1TDP1GSK3BLPLLIPG
SCHEMBL15578975 0.77 GSK3A (0.40) GSK3BLPLLIPGIRAK4
SCHEMBL392405 0.77 PRMT5 (0.47) KDM4EALDH1A1HPGDTDP1GSK3B
SCHEMBL24553447 0.76 PIM1 (0.37) NOS1ROCK2MAPTROCK1METAP2
SCHEMBL1585585 0.76 GSK3A (0.45) GSK3BLPLLIPGIRAK4KDR
SCHEMBL29644319 0.75 LPL (0.62) HIF1ALPLLIPGIRAK4
SCHEMBL1293460 0.75 LPL (0.62) HIF1ALPLLIPGIRAK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 422 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2026102082-A1 ALKYLPHENYL SUBSTITUTED COMPOUNDS, COMPOSITIONS AND METHODS OF USE DEEP APPLE THERAPEUTICS, INC. (US) 2026-05-15 WO disclosed
US-20260132119-A1 Alkylphenyl Substituted Compounds, Compositions and Methods of Use DEEP APPLE THERAPEUTICS, INC. (US) 2026-05-14 US disclosed
US-20260124222-A1 ISOTHIAZOLYLCARBOXAMIDE COMPOUNDS AND THEIR USE IN THERAPY HOTSPOT THERAPEUTICS INC (US) 2026-05-07 US disclosed
US-20260125367-A1 CANCER TREATMENTS TARGETING CANCER STEM CELLS REMEDY PLAN, INC. (US) 2026-05-07 US disclosed
EP-3886904-B1 IRAK DEGRADERS AND USES THEREOF KYMERA THERAPEUTICS INC (US) 2026-04-22 EP disclosed
US-20260092053-A1 KHK INHIBITORS GILEAD SCIENCES INC (US) 2026-04-02 US disclosed
EP-3768675-B1 NOVEL TRIAZOLONE DERIVATIVES OR SALTS THEREOF AND PHARMACEUTICAL COMPOSITIONS COMPRISING THE SAME YUHAN CORP (KR) 2026-04-01 EP disclosed
US-20260078117-A1 COMPOUNDS AND METHODS OF USE TANGO THERAPEUTICS INC (US) 2026-03-19 US disclosed
US-12577248-B2 Substituted [1,2,4]triazolo[1,5-a]pyrazines as spleen tyrosine kinase inhibitors NANJING RUIJIE PHARMA CO., LTD. (CN) 2026-03-17 US disclosed
US-20260070924-A1 INDAZOLE MACROCYCLES AND THEIR USE BLOSSOMHILL THERAPEUTICS INC (US) 2026-03-12 US disclosed
US-20080064703-A1 Fused bicycloheterocycle substituted quinuclidine derivatives ABBVIE INC. 2008-03-13 US disclosed
US-20080045539-A1 FUSED BICYCLOHETEROCYCLE SUBSTITUTED AZABICYCLIC ALKANE DERIVATIVES ABBVIE INC. 2008-02-21 US disclosed
US-20070282101-A1 Indazole compounds ABBVIE INC. 2007-12-06 US disclosed
WO-2007127175-A2 PHARMACEUTICAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2007-11-08 WO disclosed
US-20070185152-A1 Inhibitors of akt activity SMITHKLINE BEECHAM CORPORATION 2007-08-09 US disclosed
WO-2007084391-A2 THIAZOLE COMPOUNDS AS PROTEIN KINASE B ( PKB) INHIBITORS AMGEN INC. (US) 2007-07-26 WO disclosed
US-20070173506-A1 Thiazole compounds and methods of use AMGEN INC. (US) 2007-07-26 US disclosed
US-20070060588-A1 Fused bicycloheterocycle substituted quinuclidine derivatives ABBOTT LABORATORIES 2007-03-15 US disclosed
EP-1713775-A2 CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2006-10-25 EP disclosed
WO-2005074643-A2 BENZAMIDE COMPOUNDS USEFUL AS ROCK INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2005-08-18 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (13 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080045539-A1 FUSED BICYCLOHETEROCYCLE SUBSTITUTED AZABICYCLIC ALKANE DERIVATIVES MALT1, BMP2, ALKBH2 NOS1 3760/4885ROCK2 3093/4885MAPT 3978/4885
US-20070060588-A1 Fused bicycloheterocycle substituted quinuclidine derivatives CHRNA1, CHRNA7, CHRNA2 NOS1 1622/4885ROCK2 3074/4885MAPT 3296/4885
US-20070282101-A1 Indazole compounds CYP3A43, CYP3A7, UGT1A1 NOS1 849/4885ROCK2 3219/4885MAPT 2375/4885
US-20070185152-A1 Inhibitors of akt activity AKT1, AKT1S1, AKT2 NOS1 3828/4885ROCK2 713/4885MAPT 3969/4885
US-20260070924-A1 INDAZOLE MACROCYCLES AND THEIR USE NR0B2, NR0B1, ESRRA NOS1 1279/4885ROCK2 1858/4885MAPT 3932/4885
US-20080064703-A1 Fused bicycloheterocycle substituted quinuclidine derivatives IDO1, IDO2, HTR3C NOS1 1851/4885ROCK2 1550/4885MAPT 2733/4885
US-20260092053-A1 KHK INHIBITORS KHK, SLC5A2, HK1 NOS1 1762/4885ROCK2 632/4885MAPT 1585/4885
US-20070173506-A1 Thiazole compounds and methods of use MTOR, JAK2, PCK2 NOS1 2161/4885ROCK2 615/4885MAPT 2718/4885
US-20260132119-A1 Alkylphenyl Substituted Compounds, Compositions and Methods of Use GIPR, MC2R, GRPR NOS1 4219/4885ROCK2 4080/4885MAPT 4716/4885
US-20260125367-A1 CANCER TREATMENTS TARGETING CANCER STEM CELLS MCL1, MALT1, BCL6 NOS1 2646/4885ROCK2 2384/4885MAPT 4022/4885
US-20260078117-A1 COMPOUNDS AND METHODS OF USE NR3C2, ADRA1A, CNR1 NOS1 1666/4885ROCK2 1464/4885MAPT 4259/4885
US-12577248-B2 Substituted [1,2,4]triazolo[1,5-a]pyrazines as spleen tyrosine kinase inhibitors SYK, BTK, TYRO3 NOS1 1189/4885ROCK2 464/4885MAPT 2032/4885
US-20260124222-A1 ISOTHIAZOLYLCARBOXAMIDE COMPOUNDS AND THEIR USE IN THERAPY MALT1, BCL6, BCL6B NOS1 683/4885ROCK2 2950/4885MAPT 4523/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.