SCHEMBL10693674

SCHEMBL10693674

CC(C)C1(c2cccc(OCCCBr)c2)Cc2ccccc2N(C)C1=O

nearest known ligand 0.35

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 8/20 0.35
L3MBTL1 Q9Y468 2/20 0.34
GAA P10253 2/20 0.33
HSD17B10 Q99714 1/20 0.33
GRIN1 Q05586 1/20 0.33
GRIN2A Q12879 1/20 0.33
GRIN2B Q13224 1/20 0.33
BACE2 Q9Y5Z0 1/20 0.33
LMNA P02545 2/20 0.32
HTT P42858 2/20 0.32
USP2 O75604 1/20 0.32
TSHR P16473 1/20 0.32
MAPK1 P28482 1/20 0.32
ALDH1A1 P00352 1/20 0.32
DRD2 P14416 1/20 0.32
MAOA P21397 1/20 0.32
MAOB P27338 1/20 0.32
RAB9A P51151 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10692186 0.97 BACE1 (0.35) BACE1L3MBTL1GAAHSD17B10GRIN1
SCHEMBL10692789 0.89 BACE1 (0.37) BACE1GAAHSD17B10BACE2LMNA
SCHEMBL10694802 0.84 BACE1 (0.44) BACE1BACE2TSHRALDH1A1
SCHEMBL10694665 0.81 RAD52 (0.36) HSD17B10LMNAHTTTSHRALDH1A1
SCHEMBL10693819 0.77 OPRD1 (0.40)
SCHEMBL10696619 0.77 RAD52 (0.34) HSD17B10HTTALDH1A1DRD2
SCHEMBL10691593 0.74 L3MBTL1 (0.42) BACE1L3MBTL1BACE2LMNATSHR
SCHEMBL10691351 0.71 GPR55 (0.39) GAAHSD17B10LMNAHTTTSHR
SCHEMBL10674089 0.68 BACE1 (0.37) BACE1L3MBTL1GAAHSD17B10BACE2
SCHEMBL10691597 0.67 ADRA1A (0.39) L3MBTL1GAATSHRALDH1A1DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4778793-A CONTROLLING CALCIUM CONCENTRATION-CARDIOVASCULAR DISORDERS HOECHST AKTIENGESELLSCHAFT (DE) 1988-10-18 US disclosed
EP-0212216-A1 Dihydroquinolinone derivatives, processes for their preparation, medicaments containing them, the use of these medicaments, and intermediates for their preparation HOECHST AKTIENGESELLSCHAFT (DE) 1987-03-04 EP disclosed