SCHEMBL11099774

SCHEMBL11099774

CC12CCC(CCC1C(=O)O)N2Cc1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GRM6 O15303 1/20 0.40
CYP2D6 P10635 1/20 0.39
S1PR1 P21453 1/20 0.38
S1PR5 Q9H228 1/20 0.38
OPRM1 P35372 3/20 0.38
OPRK1 P41145 2/20 0.38
HSD11B1 P28845 1/20 0.38
MEN1 O00255 1/20 0.38
LMNA P02545 1/20 0.38
KMT2A Q03164 1/20 0.38
OPRD1 P41143 1/20 0.38
KCNH2 Q12809 1/20 0.38
AMPD2 Q01433 1/20 0.38
GAA P10253 1/20 0.38
SIGMAR1 Q99720 1/20 0.38
HRH3 Q9Y5N1 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1011496 0.79 HSD11B1 (0.38) CYP2D6S1PR1S1PR5HSD11B1MEN1
SCHEMBL17311985 0.72 NR1H2 (0.40) GRM6CYP2D6S1PR1S1PR5OPRM1
SCHEMBL1012463 0.72 FKBP1A (0.45) KMT2A
SCHEMBL10202890 0.71 ALDH1A1 (0.60) CYP2D6S1PR1S1PR5OPRM1OPRK1
SCHEMBL11093783 0.69 CCR2 (0.41) CYP2D6OPRK1HSD11B1AMPD2GAA
SCHEMBL22443390 0.68 GRM6 (0.51) GRM6CYP2D6S1PR1S1PR5OPRK1
SCHEMBL1203078 0.68 DRD2 (0.41) OPRK1HSD11B1MEN1LMNAKMT2A
Hydrochloric Acid SCHEMBL9837514 0.68 KMT2A (0.40) CYP2D6OPRK1MEN1LMNAKMT2A
SCHEMBL1012462 0.68 HSD11B1 (0.40) CYP2D6OPRM1HSD11B1MEN1KMT2A
SCHEMBL3250253 0.67 OPRK1 (0.51) OPRK1SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0031219-B1 ANILINE DERIVATIVES BEECHAM GROUP PLC (GB) 1984-03-07 EP disclosed
US-4350691-A ANTIEMETICS BEECHAM GROUP LIMITED (GB) 1982-09-21 US disclosed
EP-0031219-A1 Aniline derivatives BEECHAM GROUP PLC (GB) 1981-07-01 EP disclosed