SCHEMBL1141383

SCHEMBL1141383

CC(C)(C)OC(=O)NCCc1ccc(B2OC(C)(C)C(C)(C)O2)cc1

nearest known ligand 0.70

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CA2 P00918 4/20 0.55
CA1 P00915 3/20 0.55
CA9 Q16790 2/20 0.55
AAK1 Q2M2I8 2/20 0.52
PRMT5 O14744 1/20 0.51
WDR77 Q9BQA1 1/20 0.51
LPL P06858 5/20 0.50
LIPG Q9Y5X9 5/20 0.50
NAMPT P43490 1/20 0.47
F11 P03951 2/20 0.46
F2 P00734 1/20 0.46
PRSS1 P07477 1/20 0.46
PRSS2 P07478 1/20 0.46
PRSS3 P35030 1/20 0.46
MAPT P10636 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
LMNA P02545 1/20 0.42
DGAT1 O75907 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16947897 0.93 LPL (0.51) CA2CA1CA9AAK1PRMT5
SCHEMBL15585542 0.92 CA2 (0.50) CA2CA1CA9AAK1PRMT5
SCHEMBL22767308 0.92 LPL (0.53) CA2CA1CA9AAK1PRMT5
SCHEMBL16169739 0.88 PRMT5 (0.48) CA2CA1CA9AAK1PRMT5
SCHEMBL169651 0.87 PRMT5 (0.58) CA2CA1CA9AAK1PRMT5
SCHEMBL2144320 0.86 LIPG (0.51) CA2CA1CA9AAK1PRMT5
SCHEMBL1990625 0.84 CA1 (0.54) CA2CA1CA9AAK1PRMT5
SCHEMBL15805934 0.83 PRMT5 (0.46) CA2CA1CA9AAK1PRMT5
SCHEMBL15919266 0.83 AAK1 (0.61) CA2CA1CA9AAK1PRMT5
SCHEMBL16947773 0.82 DGAT1 (0.50) CA2CA1CA9AAK1PRMT5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 126 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2970176-B1 MOLECULES HAVING CERTAIN PESTICIDAL UTILITIES, AND INTERMEDIATES, COMPOSITIONS, AND PROCESSES RELATED THERETO CORTEVA AGRISCIENCE LLC (US) 2023-10-25 EP disclosed
EP-2970176-B1 MOLECULES HAVING CERTAIN PESTICIDAL UTILITIES, AND INTERMEDIATES, COMPOSITIONS, AND PROCESSES RELATED THERETO CORTEVA AGRISCIENCE LLC (US) 2023-10-25 EP disclosed
WO-2023153504-A1 NUCLEIC ACID DELIVERY MATERIAL 国立大学法人東海国立大学機構 2023-08-17 WO disclosed
US-20230167073-A1 ARYL OR HETEROARYL DERIVATIVE TEIJIN PHARMA LIMITED (JP) 2023-06-01 US disclosed
CN-115996910-A Aryl or heteroaryl derivatives 帝人制药株式会社 2023-04-21 CN disclosed
EP-4137481-A1 ARYL OR HETEROARYL DERIVATIVE Teijin Pharma Limited (JP) 2023-02-22 EP disclosed
US-20230029009-A1 CHEMICAL COMPOUNDS BLUE OWL CAPITAL CORPORATION, AS NEW AGENT 2023-01-26 US disclosed
US-20230029009-A1 CHEMICAL COMPOUNDS BLUE OWL CAPITAL CORPORATION, AS NEW AGENT 2023-01-26 US disclosed
US-11459331-B2 Chemical compounds AVISTA PHARMA SOLUTIONS, INC. (US) 2022-10-04 US disclosed
EP-4026832-A1 PIPERIDINE DERIVATIVES AS INHIBITORS OF UBIQUITIN SPECIFIC PROTEASE 7 Almac Discovery Limited (GB) 2022-07-13 EP disclosed
US-20090318436-A1 Fused heterocyclic derivatives and methods of use AMGEN INC. (US) 2009-12-24 US disclosed
US-20090264468-A1 Methods for treating a disease in which Rho kinase is involved UBE INDUSTRIES, LTD. (JP) 2009-10-22 US disclosed
WO-2009091374-A2 FUSED HETEROCYCLIC DERIVATIVES AND METHODS OF USE AMGEN INC. (US) 2009-07-23 WO disclosed
WO-2009091374-A2 FUSED HETEROCYCLIC DERIVATIVES AND METHODS OF USE AMGEN INC. (US) 2009-07-23 WO disclosed
US-7563906-B2 Indazole derivatives UBE INDUSTRIES, LTD. (JP) 2009-07-21 US disclosed
US-20090124609-A1 Fused heterocyclic derivatives and methods of use AMGEN INC. (US) 2009-05-14 US disclosed
US-20090124609-A1 Fused heterocyclic derivatives and methods of use AMGEN INC. (US) 2009-05-14 US disclosed
US-20090124609-A1 Fused heterocyclic derivatives and methods of use AMGEN INC. (US) 2009-05-14 US disclosed
US-20070129404-A1 Novel indazole derivatives UBE INDUSTRIES, LTD. (JP) 2007-06-07 US disclosed
EP-1679308-A1 NOVEL INDAZOLE DERIVATIVE Ube Industries, Ltd. (JP) 2006-07-12 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090318436-A1 Fused heterocyclic derivatives and methods of use HGF, HGFAC, MET CA2 3345/4885CA1 2847/4885CA9 1334/4885
US-20230167073-A1 ARYL OR HETEROARYL DERIVATIVE ARRB1, NR3C2, TRPC6 CA2 2861/4885CA1 4852/4885CA9 4469/4885
US-11459331-B2 Chemical compounds PTGER4, PTGES, PTGES2 CA2 2133/4885CA1 4486/4885CA9 3503/4885
US-20230029009-A1 CHEMICAL COMPOUNDS PTGER4, PTGES, PTGES2 CA2 2133/4885CA1 4486/4885CA9 3503/4885
US-20090264468-A1 Methods for treating a disease in which Rho kinase is involved RHOA, ROCK1, RHOT2 CA2 743/4885CA1 3375/4885CA9 3299/4885
US-20070129404-A1 Novel indazole derivatives CIT, ROCK1, ROCK2 CA2 1567/4885CA1 4768/4885CA9 4437/4885
US-20090124609-A1 Fused heterocyclic derivatives and methods of use HGF, HGFAC, MET CA2 3345/4885CA1 2847/4885CA9 1334/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.