SCHEMBL12413657

SCHEMBL12413657

CC(C)C(=O)NCCC1CCNCC1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 2/20 0.57
ITGB3 P05106 5/20 0.44
ITGA2B P08514 5/20 0.44
TPSAB1 Q15661 1/20 0.44
TPSD1 Q9BZJ3 1/20 0.44
TPSG1 Q9NRR2 1/20 0.44
BCHE P06276 1/20 0.42
ALOX15 P16050 2/20 0.41
CHRM1 P11229 2/20 0.40
CHRM2 P08172 1/20 0.40
CHRM3 P20309 1/20 0.40
NQO2 P16083 1/20 0.39
MTNR1A P48039 1/20 0.39
MTNR1B P49286 1/20 0.39
PRMT3 O60678 1/20 0.38
TSHR P16473 1/20 0.38
NAMPT P43490 1/20 0.38
ROCK2 O75116 1/20 0.38
EPHX1 P07099 1/20 0.37
CPN1 P15169 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11090 0.87 SIGMAR1 (0.49) SIGMAR1BCHENQO2MTNR1AMTNR1B
SCHEMBL24276406 0.84 SIGMAR1 (0.57) SIGMAR1BCHENQO2MTNR1AMTNR1B
SCHEMBL10446115 0.82 ALOX15 (0.54) SIGMAR1ALOX15CHRM1TSHREPHX1
SCHEMBL9891794 0.82 SIGMAR1 (0.60) SIGMAR1BCHENQO2MTNR1AMTNR1B
SCHEMBL1037980 0.80 ALOX15 (0.47) SIGMAR1ITGB3ITGA2BTPSAB1TPSD1
SCHEMBL9891910 0.79 SIGMAR1 (0.43) SIGMAR1BCHENQO2MTNR1AMTNR1B
Hydrochloric Acid SCHEMBL7417264 0.79 ALOX15 (0.46) SIGMAR1ITGB3ITGA2BTPSAB1TPSD1
SCHEMBL16011477 0.79 ITGB3 (0.46) SIGMAR1ITGB3ITGA2BTPSAB1TPSD1
SCHEMBL1290747 0.78 ITGB3 (0.51) SIGMAR1ITGB3ITGA2BTPSAB1TPSD1
SCHEMBL23168317 0.78 GNAI3 (0.44) SIGMAR1CHRM1EPHX1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024026484-A2 CDK2 INHIBITORS AND METHODS OF USING THE SAME CEDILLA THERAPEUTICS, INC. (US) 2024-02-01 WO disclosed
US-10428080-B2 TBK/IKK inhibitor compounds and uses thereof MERCK PATENT GMBH (DE) 2019-10-01 US disclosed
US-9988391-B2 TBK/IKK inhibitor compounds and uses thereof MERCK PATENT GMBH (DE) 2018-06-05 US disclosed
US-9988391-B2 TBK/IKK inhibitor compounds and uses thereof MERCK PATENT GMBH (DE) 2018-06-05 US disclosed
US-8293729-B2 Compounds, pharmaceutical composition and methods relating thereto BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-10-23 US disclosed
US-8293729-B2 Compounds, pharmaceutical composition and methods relating thereto BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-10-23 US disclosed
US-20110166116-A1 NEW COMPOUNDS, PHARMACEUTICAL COMPOSITION AND METHODS RELATING THERETO BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2011-07-07 US disclosed
US-20110166116-A1 NEW COMPOUNDS, PHARMACEUTICAL COMPOSITION AND METHODS RELATING THERETO BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2011-07-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10428080-B2 TBK/IKK inhibitor compounds and uses thereof NFKBIA, TBKBP1, TBK1 SIGMAR1 4797/4885ITGB3 2218/4885ITGA2B 2204/4885
US-20110166116-A1 NEW COMPOUNDS, PHARMACEUTICAL COMPOSITION AND METHODS RELATING THERETO MC2R, REN, CYP11B2 SIGMAR1 1562/4885ITGB3 3653/4885ITGA2B 4274/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.