SCHEMBL13628860

SCHEMBL13628860

COOSc1ccc2c(c1)cc(-c1cc[n+]([O-])cc1)n2Cc1ccc(F)cc1

nearest known ligand 0.46

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 4/20 0.46
TP53 P04637 1/20 0.32
MAPT P10636 1/20 0.32
LMNA P02545 1/20 0.32
GRIK1 P39086 1/20 0.32
GRIK2 Q13002 1/20 0.32
TBXA2R P21731 1/20 0.32
GNRHR P30968 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13628848 0.89 PTGS2 (0.42) PTGS2LMNAGRIK1GRIK2GNRHR
SCHEMBL13628859 0.85 PTGS2 (0.45) PTGS2TP53TBXA2RGNRHR
SCHEMBL13628847 0.80 CYP11B2 (0.43) PTGS2MAPTGNRHR
SCHEMBL2922397 0.79 PTGS2 (0.66) PTGS2TBXA2RGNRHR
SCHEMBL13628821 0.78 MAPT (0.37) PTGS2TP53MAPTLMNATBXA2R
SCHEMBL13628832 0.78 TRPC5 (0.38) PTGS2MAPT
SCHEMBL13628853 0.77 PTGS2 (0.37) PTGS2MAPTLMNATBXA2R
SCHEMBL13628851 0.76 PTGS2 (0.36) PTGS2TP53TBXA2R
SCHEMBL13628824 0.76 RAB9A (0.36) PTGS2MAPTTBXA2R
SCHEMBL13628850 0.76 PTGS2 (0.36) PTGS2MAPTLMNATBXA2R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7612070-B2 Heterocyclic compounds as antiinflammatory agents and cyclooxygenase inhibitors CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2009-11-03 US disclosed