SCHEMBL13717271

SCHEMBL13717271

CCCCC(C#N)C(=O)[O-].[Na+]

nearest known ligand 0.52

Known targets — ChEMBL curated mechanism

ABCC8ACEADORA1ADORA2AADORA2BADORA3ALDH5A1ALOX5ALOX5APATP4AATP4BBRAFCA1CA12CA2CA4CYSLTR1DHFRDPEP1EDNRAEDNRBESR2F10FDPSFGF1GABBR1GABBR2GABRA1GABRA2GABRA3GABRA4GABRA5GABRA6GABRB1GABRB2GABRB3GABRDGABREGABRG1GABRG2GABRG3GABRPGABRQGARTGNRHRGSC1HMGCRIMPDH1IMPDH2KCNJ11LY96NOD2NR3C1NS3NS4ANS5bP2RY1P2RY12P2RY2P2RY4P2RY6PBP2XPDE3APDE3BPDE4APDE4BPDE4CPDE4DPDK1PDK2PDK3PDK4PPARGPPATPTGIRPTGS1PTGS2RAF1RYR1RYR3SCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASERPINC1SLC12A1SLC12A3SYKTHRATHRBTLR3TLR4TLR9TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYMSVKORC1XDHblablaIMP-1blaOXA-33blaOXA-58blaT-3blaT-4blaT-5blaT-6dacAdacBdacCfolAfolPfolP1ftsIfusAgaggyrAgyrBmecAmrcAmrcBmrdApbp1apbp1bpbp2pbp2apbp2bpbp3pbp4pbpApbpBpbpCpbpFpolponBrplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpoArpoBrpoCrpoZrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of None. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CA2 known ✓ P00918 6/20 0.52
CA1 known ✓ P00915 4/20 0.47
NFKB1 P19838 3/20 0.43
TSHR P16473 3/20 0.43
CYP3A4 P08684 2/20 0.43
NPSR1 Q6W5P4 2/20 0.43
GPR84 Q9NQS5 1/20 0.38
MAPK1 P28482 1/20 0.36
CES1 P23141 2/20 0.35
CES2 O00748 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL316535 0.79 CA2 (0.48) CA2CA1TSHRGPR84MAPK1
SCHEMBL10627769 0.79 CA2 (0.39) CA2CA1TSHRGPR84MAPK1
SCHEMBL16016004 0.79 CA2 (0.39) CA2CA1TSHRGPR84MAPK1
SCHEMBL10591035 0.79
SCHEMBL319447 0.78 CA2 (0.50) CA2CA1TSHRMAPK1
SCHEMBL4338848 0.78 CA1 (0.45) CA2CA1NFKB1TSHRCYP3A4
SCHEMBL16006551 0.78 ALDH1A1 (0.38) CA2CA1TSHRGPR84MAPK1
SCHEMBL10748206 0.77 CA2 (0.42) CA2CA1NFKB1GPR84
SCHEMBL10627704 0.76 CA2 (0.36) CA2CA1TSHRMAPK1CES1
SCHEMBL9562158 0.74 CA2 (0.40) CA2CA1TSHRCYP3A4MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8651185-B2 Reducing or stopping the uncontrolled flow of fluid such as oil from a well LOS ALAMOS NATIONAL SECURITY, LLC (US) 2014-02-18 US claimed
US-20120285683-A1 REDUCING OR STOPPING THE UNCONTROLLED FLOW OF FLUID SUCH AS OIL FROM A WELL LOS ALAMOS NATIONAL SECURITY, LLC (US) 2012-11-15 US claimed
US-8651185-B2 Reducing or stopping the uncontrolled flow of fluid such as oil from a well LOS ALAMOS NATIONAL SECURITY, LLC (US) 2014-02-18 US disclosed
US-20120285683-A1 REDUCING OR STOPPING THE UNCONTROLLED FLOW OF FLUID SUCH AS OIL FROM A WELL LOS ALAMOS NATIONAL SECURITY, LLC (US) 2012-11-15 US disclosed