SCHEMBL144836

SCHEMBL144836

CC(=O)C1(NC(=O)OC(C)(C)C)CC1

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
MAPK1 P28482 1/20 0.39
GHSR Q92847 1/20 0.36
CTSL P07711 1/20 0.35
APLNR P35414 1/20 0.35
TDP1 Q9NUW8 1/20 0.34
NFKB1 P19838 1/20 0.34
NFKB2 Q00653 1/20 0.34
RELA Q04206 1/20 0.34
GAA P10253 4/20 0.33
DGAT1 O75907 1/20 0.33
BTK Q06187 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA7 P43166 1/20 0.33
CTSK P43235 1/20 0.33
RORC P51449 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12175055 0.92 MEN1 (0.37) MEN1KMT2AMAPK1GHSRCTSL
SCHEMBL2712148 0.92 MEN1 (0.37) MEN1KMT2AMAPK1GHSRCTSL
SCHEMBL15116717 0.91 TSHR (0.37) MEN1KMT2AMAPK1GHSRCTSL
SCHEMBL15116645 0.91 GAA (0.36) MEN1KMT2AMAPK1GHSRCTSL
SCHEMBL15116541 0.88 USP2 (0.38) MEN1KMT2AMAPK1GHSRCTSL
SCHEMBL16409146 0.86 GHSR (0.39) MEN1KMT2AMAPK1GHSRCTSL
SCHEMBL142219 0.84 MEN1 (0.39) MEN1KMT2AMAPK1GHSRCTSL
SCHEMBL15116710 0.83 GAA (0.43) MEN1KMT2AMAPK1GHSRAPLNR
SCHEMBL2392486 0.82 KMT2A (0.38) MEN1KMT2AMAPK1GHSRCTSL
SCHEMBL1820679 0.82 MAPT (0.39) MEN1KMT2AMAPK1GHSRCTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 34 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230201353-A1 SUSTAINED RELEASE DELIVERY SYSTEMS COMPRISING TRACELESS LINKERS NOVARTIS AG (CH) 2023-06-29 US disclosed
CN-110997661-B Cyclopropyl ureaplatin 2 receptor and formyl peptide 1 receptor agonists 百时美施贵宝公司 2023-03-31 CN disclosed
US-20220323595-A1 SUSTAINED DELIVERY OF ANGIOPOETIN-LIKE 3 POLYPEPTIDES NOVARTIS AG (CH) 2022-10-13 US disclosed
US-11180490-B2 Cyclopropyl urea formyl peptide 2 receptor and formyl peptide 1 receptor agonists BRISTOL-MYERS SQUIBB COMPANY (US) 2021-11-23 US disclosed
EP-3634958-B1 CYCLOPROPYL UREA FORMYL PEPTIDE 2 RECEPTOR AND FORMYL PEPTIDE 1 RECEPTOR AGONISTS BRISTOL MYERS SQUIBB CO (US) 2021-07-21 EP disclosed
WO-2021050612-A1 COMPOSITIONS AND METHODS FOR THE TREATMENT OF RESPIRATORY SYNCYTIAL VIRUS CIDARA THERAPEUTICS, INC. (US) 2021-03-18 WO disclosed
US-20200376129-A1 SUSTAINED RELEASE DELIVERY SYSTEMS COMPRISING TRACELESS LINKERS NOVARTIS INSTITUTES FOR BIOMEDICAL RESEARCH, INC. 2020-12-03 US disclosed
US-10751417-B2 Sustained release delivery systems comprising traceless linkers NOVARTIS AG (CH) 2020-08-25 US disclosed
US-20200199113-A1 CYCLOPROPYL UREA FORMYL PEPTIDE 2 RECEPTOR AND FORMYL PEPTIDE 1 RECEPTOR AGONISTS BRISTOL MYERS SQUIBB CO (US) 2020-06-25 US disclosed
CN-110997661-A Cyclopropyl ureaplatin 2 receptor and formyl peptide 1 receptor agonists 百时美施贵宝公司 2020-04-10 CN disclosed
US-8354410-B2 Compounds for the treatment of hepatitis C BRISTOL-MEYERS SQUIBB COMPANY (US) 2013-01-15 US disclosed
US-8354410-B2 Compounds for the treatment of hepatitis C BRISTOL-MEYERS SQUIBB COMPANY (US) 2013-01-15 US disclosed
US-20120059019-A1 Compounds for the Treatment of Hepatitis C BRISTOL-MYERS SQUIBB COMPANY 2012-03-08 US disclosed
US-20120059019-A1 Compounds for the Treatment of Hepatitis C BRISTOL-MYERS SQUIBB COMPANY 2012-03-08 US disclosed
WO-2011112769-A1 COMPOUNDS FOR THE TREATMENT OF HEPATITIS C BRISTOL-MYERS SQUIBB COMPANY (US) 2011-09-15 WO disclosed
WO-2011112769-A1 COMPOUNDS FOR THE TREATMENT OF HEPATITIS C BRISTOL-MYERS SQUIBB COMPANY (US) 2011-09-15 WO disclosed
US-20110224188-A1 DERIVATIVES OF 6,7-DIHYDRO-5H-IMIDAZO[1,2-alpha]IMIDAZOLE-3-CARBOXYLIC ACID AMIDES BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2011-09-15 US disclosed
US-20090156572-A1 Nitrogen-containing heterocyclic compound and use thereof TAKEDA PHARMACEUTICAL COMPANY LIMITED 2009-06-18 US disclosed
US-20090156572-A1 Nitrogen-containing heterocyclic compound and use thereof TAKEDA PHARMACEUTICAL COMPANY LIMITED 2009-06-18 US disclosed
WO-2009070485-A1 DERIVATIVES OF 6,7-DIHYDRO-5H-IMIDAZO[1,2-α]IMIDAZOLE-3- CARBOXYLIC ACID AMIDES BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2009-06-04 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (9 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110224188-A1 DERIVATIVES OF 6,7-DIHYDRO-5H-IMIDAZO[1,2-alpha]IMIDAZOLE-3-CARBOXYLIC ACID AMIDES HPGDS, COL14A1, ARG1 MEN1 4830/4885KMT2A 2995/4885MAPK1 1413/4885
US-11180490-B2 Cyclopropyl urea formyl peptide 2 receptor and formyl peptide 1 receptor agonists FPR1, FPR2, FPR3 MEN1 4563/4885KMT2A 4752/4885MAPK1 958/4885
US-20230201353-A1 SUSTAINED RELEASE DELIVERY SYSTEMS COMPRISING TRACELESS LINKERS ABCB11, ABCB1, GHRHR MEN1 2713/4885KMT2A 1725/4885MAPK1 2336/4885
US-20200376129-A1 SUSTAINED RELEASE DELIVERY SYSTEMS COMPRISING TRACELESS LINKERS ABCB11, ABCB1, GHRHR MEN1 2713/4885KMT2A 1725/4885MAPK1 2336/4885
US-20120059019-A1 Compounds for the Treatment of Hepatitis C HAVCR2, HCCS, SLC10A1 MEN1 4676/4885KMT2A 4624/4885MAPK1 3142/4885
US-10751417-B2 Sustained release delivery systems comprising traceless linkers ABCB11, ABCB1, GHRHR MEN1 2713/4885KMT2A 1725/4885MAPK1 2336/4885
US-20200199113-A1 CYCLOPROPYL UREA FORMYL PEPTIDE 2 RECEPTOR AND FORMYL PEPTIDE 1 RECEPTOR AGONISTS FPR1, FPR2, FPR3 MEN1 4563/4885KMT2A 4752/4885MAPK1 958/4885
US-20220323595-A1 SUSTAINED DELIVERY OF ANGIOPOETIN-LIKE 3 POLYPEPTIDES TEK, VEGFA, FLT4 MEN1 695/4885KMT2A 3702/4885MAPK1 3278/4885
US-20090156572-A1 Nitrogen-containing heterocyclic compound and use thereof NTSR2, NTSR1, HNMT MEN1 206/4885KMT2A 977/4885MAPK1 1405/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.