SCHEMBL1532393

SCHEMBL1532393

O=c1nc[nH]c2c1ncn2[C@@H]1O[C@H](COP(=O)([O-])[O-])[C@@H](O)[C@H]1O.[Na+].[Na+]

nearest known ligand 0.57

Known targets — ChEMBL curated mechanism

ABCC8ACEADORA1ADORA2AADORA2BADORA3ALDH5A1ALOX5ALOX5APATP4AATP4BBRAFCA1CA12CA2CA4CYSLTR1DHFRDPEP1EDNRAEDNRBESR2F10FDPSFGF1GABBR1GABBR2GABRA1GABRA2GABRA3GABRA4GABRA5GABRA6GABRB1GABRB2GABRB3GABRDGABREGABRG1GABRG2GABRG3GABRPGABRQGARTGNRHRGSC1HMGCRIMPDH1IMPDH2KCNJ11LY96NOD2NR3C1NS3NS4ANS5bP2RY1P2RY12P2RY2P2RY4P2RY6PBP2XPDE3APDE3BPDE4APDE4BPDE4CPDE4DPDK1PDK2PDK3PDK4PPARGPPATPTGIRPTGS1PTGS2RAF1RYR1RYR3SCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASERPINC1SLC12A1SLC12A3SYKTHRATHRBTLR3TLR4TLR9TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYMSVKORC1XDHblablaIMP-1blaOXA-33blaOXA-58blaT-3blaT-4blaT-5blaT-6dacAdacBdacCfolAfolPfolP1ftsIfusAgaggyrAgyrBmecAmrcAmrcBmrdApbp1apbp1bpbp2pbp2apbp2bpbp3pbp4pbpApbpBpbpCpbpFpolponBrplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpoArpoBrpoCrpoZrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of None. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA1 known ✓ P30542 3/20 0.52
P2RY1 known ✓ P47900 6/20 0.52
ADORA3 known ✓ P0DMS8 1/20 0.50
ADORA2A known ✓ P29274 1/20 0.50
IMPDH2 known ✓ P12268 5/20 0.48
IMPDH1 known ✓ P20839 1/20 0.48
P2RY2 known ✓ P41231 1/20 0.48
PDE4D known ✓ Q08499 1/20 0.48
PDE3A known ✓ Q14432 1/20 0.48
P2RY12 known ✓ Q9H244 1/20 0.47
P2RX3 P56373 1/20 0.57
ENPP1 P22413 2/20 0.52
P2RY11 Q96G91 3/20 0.49
DNPH1 O43598 1/20 0.48
PRKAB2 O43741 1/20 0.48
TRPM2 O94759 1/20 0.48
LDHA P00338 1/20 0.48
ADRB2 P07550 1/20 0.48
FBP1 P09467 1/20 0.48
SRC P12931 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL316942 1.00 P2RX3 (0.57) P2RX3ADORA1P2RY1ENPP1ADORA3
SCHEMBL1030880 0.99 P2RX3 (0.56) P2RX3ADORA1P2RY1ENPP1ADORA3
Water SCHEMBL20266269 0.99 P2RX3 (0.56) P2RX3ADORA1P2RY1ENPP1ADORA3
SCHEMBL2683124 0.91 P2RX3 (0.61) P2RX3ADORA1P2RY1P2RY11IMPDH2
SCHEMBL184241 0.91 P2RX3 (0.61) P2RX3ADORA1P2RY1P2RY11IMPDH2
SCHEMBL4356525 0.87 P2RX3 (0.67) P2RX3P2RY1ENPP1P2RY11TRPM2
SCHEMBL4368535 0.87 P2RX3 (0.67) P2RX3P2RY1ENPP1P2RY11TRPM2
SCHEMBL24059927 0.85 P2RX3 (0.70) P2RX3P2RY1ENPP1P2RY11TRPM2
SCHEMBL4356292 0.85 P2RX3 (0.70) P2RX3P2RY1ENPP1P2RY11TRPM2
SCHEMBL4363134 0.85 P2RX3 (0.70) P2RX3P2RY1ENPP1P2RY11TRPM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 18 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4630407-A1 2-METHYL-2-(1-METHYLCYCLOHEXYL)PROPANAMIDE DERIVATIVES AND 1-(TERT-BUTYL)-CYCLOHEXANE-1-CARBOXAMIDE DERIVATIVES FOR USE IN UMAMI FLAVOR COMPOSITIONS International Flavors & Fragrances, Inc. (US) 2025-10-15 EP disclosed
CN-118125875-B Amino acid-containing water-soluble fertilizer and preparation method thereof 广州市绿量有机肥料有限公司 2024-11-29 CN disclosed
CN-118125875-A Amino acid-containing water-soluble fertilizer and preparation method thereof 广州市绿量有机肥料有限公司 2024-06-04 CN disclosed
US-11612575-B2 Combination therapies with disulfiram Spring Discovery, Inc. (US) 2023-03-28 US disclosed
US-20220087956-A1 COMBINATION THERAPIES WITH DISULFIRAM WINTER ACQUISITION SUB, INC. 2022-03-24 US disclosed
US-20220087955-A1 COMBINATION THERAPIES WITH DISULFIRAM WINTER ACQUISITION SUB, INC. 2022-03-24 US disclosed
US-11065214-B1 Combination therapies with disulfiram Spring Discovery, Inc. (US) 2021-07-20 US disclosed
CN-110074399-A For promoting the alimentation composition of satiety MJN 美国控股有限责任公司 2019-08-02 CN disclosed
CN-106999973-A System and method for discharging edible material 阿甘芳香和精细化工有限公司 2017-08-01 CN disclosed
EP-2292585-B1 Screening for solid forms by ultrasound crystallization and cocrystallization using ultrasound APTUIT WEST LAFAYETTE LLC (US) 2016-04-27 EP disclosed
EP-2931064-A1 NUTRITIONAL COMPOSITION FOR PROMOTING SATIETY MJN U.S. Holdings, LLC (US) 2015-10-21 EP disclosed
CN-104837368-A Nutritional composition for promoting satiety MJN US HOLDINGS LLC 2015-08-12 CN disclosed
US-8920559-B2 Screening for solid forms by ultrasound crystallization and cocrystallization using ultrasound APTUIT (WEST LAFAYETTE), LLC (US) 2014-12-30 US disclosed
WO-2014092861-A1 NUTRITIONAL COMPOSITION FOR PROMOTING SATIETY MJN U.S. HOLDINGS LLC (US) 2014-06-19 WO disclosed
US-20140170259-A1 NUTRITIONAL COMPOSITION FOR PROMOTING SATIETY MEAD JOHNSON NUTRITION COMPANY (US) 2014-06-19 US disclosed
US-20110257430-A1 NOVEL COCRYSTALLIZATION APTUIT (KANSAS CITY), LLC (US) 2011-10-20 US disclosed
US-20110251426-A1 SCREENING FOR SOLID FORMS BY ULTRASOUND CRYSTALLIZATION AND COCRYSTALLIZATION USING ULTRASOUND S.S.C.I., INC. (US) 2011-10-13 US disclosed
EP-2292585-A1 Screening for solid forms by ultrasound crystallization and cocrystallization using ultrasound APTUIT (KANSAS CITY), LLC (US) 2011-03-09 EP disclosed