SCHEMBL16048397

SCHEMBL16048397

O=C(O)c1cnc(NC2CCOCC2)cn1

nearest known ligand 0.49

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HCAR3 P49019 3/20 0.49
HDAC3 O15379 1/20 0.47
HDAC1 Q13547 1/20 0.47
HDAC2 Q92769 1/20 0.47
HDAC6 Q9UBN7 1/20 0.47
CCNE1 P24864 5/20 0.46
CDK2 P24941 5/20 0.46
MAPK1 P28482 7/20 0.43
MAPK3 P27361 2/20 0.41
FYN P06241 2/20 0.41
PCSK9 Q8NBP7 1/20 0.39
MKNK1 Q9BUB5 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29582918 1.00 HCAR3 (0.49) HCAR3HDAC3HDAC1HDAC2HDAC6
SCHEMBL17075516 0.98 HCAR3 (0.48) HCAR3HDAC3HDAC1HDAC2HDAC6
SCHEMBL29944834 0.90 HDAC3 (0.46) HCAR3HDAC3HDAC1HDAC2HDAC6
SCHEMBL2817349 0.90 HDAC3 (0.46) HCAR3HDAC3HDAC1HDAC2HDAC6
Lithium Ion SCHEMBL17075514 0.85 HDAC3 (0.45) HCAR3HDAC3HDAC1HDAC2HDAC6
Fumaric Acid SCHEMBL30856933 0.85 HCAR3 (0.42) HCAR3HDAC3HDAC1HDAC2HDAC6
SCHEMBL2790974 0.84 PCSK9 (0.56) HDAC3HDAC1HDAC2HDAC6CCNE1
SCHEMBL25387892 0.78 S1PR1 (0.48) CCNE1CDK2
SCHEMBL30000505 0.78 S1PR1 (0.48) CCNE1CDK2
SCHEMBL15511812 0.76 CCNE1 (0.72) HCAR3CCNE1CDK2MAPK1MAPK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 20 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230110165-A1 Substituted Imidazo[4,5-c]pyridine Compounds and Compositions Thereof PROXIMAGEN LLC (US) 2023-04-13 US disclosed
US-10968223-B2 Imidazo[4,5-c]pyridine and pyrrolo[2,3-c]pyridine derivatives as SSAO inhibitors PROXIMAGEN, LLC (US) 2021-04-06 US disclosed
US-20200347059-A1 IMIDAZO[4,5-C]PYRIDINE AND PYRROLO[2,3-C]PYRIDINE DERIVATIVES AS SSAO INHIBITORS PROXIMAGEN, LLC (US) 2020-11-05 US disclosed
US-10766897-B2 Imidazo[4,5-c]pyridine and pyrrolo[2,3-c]pyridine derivatives as SSAO inhibitors PROXIMAGEN, LLC (US) 2020-09-08 US disclosed
US-20200262835-A1 COMPOUNDS PROXIMAGEN, LLC (US) 2020-08-20 US disclosed
US-10590125-B2 Compounds PROXIMAGEN, LLC (US) 2020-03-17 US disclosed
US-10428066-B2 Imidazo[4,5-C]pyridine and pyrrolo[2,3-C]pyridine derivatives as SSAO inhibitors PROXIMAGEN, LLC (US) 2019-10-01 US disclosed
EP-2970260-B1 IMIDAZO[4,5-C]PYRIDINE AND PYRROLO[2,3-C]PYRIDINE DERIVATIVES AS SSAO INHIBITORS PROXIMAGEN LLC (US) 2019-04-24 EP disclosed
US-20180194763-A1 IMIDAZO[4,5-C]PYRIDINE AND PYRROLO[2,3-C]PYRIDINE DERIVATIVES AS SSAO INHIBITORS PROXIMAGEN LIMITED (GB) 2018-07-12 US disclosed
US-9951068-B2 Imidazo[4,5-C]pyridine and pyrrolo[2,3-C]pyridine derivatives as SSAO inhibitors PROXIMAGEN LIMITED (GB) 2018-04-24 US disclosed
US-20170247378-A1 IMIDAZO[4,5-C]PYRIDINE AND PYRROLO[2,3-C]PYRIDINE DERIVATIVES AS SSAO INHIBITORS PROXIMAGEN, LLC 2017-08-31 US disclosed
US-9676769-B2 Imidazo[4,5-C]pyridine and pyrrolo[2,3-C]pyridine derivatives as SSAO inhibitors PROXIMAGEN LIMITED (GB) 2017-06-13 US disclosed
US-20160326172-A1 NEW COMPOUNDS PROXIMAGEN, LLC 2016-11-10 US disclosed
US-20160326172-A1 NEW COMPOUNDS PROXIMAGEN, LLC 2016-11-10 US disclosed
US-9428498-B2 Substituted imidazo[4,5-c]pyridine compounds and compositions thereof PROXIMAGEN LIMITED (GB) 2016-08-30 US disclosed
US-9428498-B2 Substituted imidazo[4,5-c]pyridine compounds and compositions thereof PROXIMAGEN LIMITED (GB) 2016-08-30 US disclosed
US-20150258101-A1 NEW COMPOUNDS PROXIMAGEN LIMITED (GB) 2015-09-17 US disclosed
WO-2014140592-A1 IMIDAZO[4,5-C]PYRIDINE AND PYRROLO[2,3-C]PYRIDINE DERIVATIVES AS SSAO INHIBITORS PROXIMAGEN LIMITED (GB) 2014-09-18 WO disclosed
US-20140275040-A1 NEW COMPOUNDS PROXIMAGEN LIMITED (GB) 2014-09-18 US disclosed
US-20140275040-A1 NEW COMPOUNDS PROXIMAGEN LIMITED (GB) 2014-09-18 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (12 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10590125-B2 Compounds ALOX15B, ALOX12, ALOX15 HCAR3 660/4885HDAC3 2894/4885HDAC1 1649/4885
US-20160326172-A1 NEW COMPOUNDS SSB, ALOX15B, ALOX12 HCAR3 511/4885HDAC3 3108/4885HDAC1 1874/4885
US-10766897-B2 Imidazo[4,5-c]pyridine and pyrrolo[2,3-c]pyridine derivatives as SSAO inhibitors PNPO, SSB, XDH HCAR3 1797/4885HDAC3 1948/4885HDAC1 699/4885
US-10428066-B2 Imidazo[4,5-C]pyridine and pyrrolo[2,3-C]pyridine derivatives as SSAO inhibitors PNPO, SSB, XDH HCAR3 1797/4885HDAC3 1948/4885HDAC1 699/4885
US-20140275040-A1 NEW COMPOUNDS SSB, ALOX15B, ALOX12 HCAR3 511/4885HDAC3 3108/4885HDAC1 1874/4885
US-20170247378-A1 IMIDAZO[4,5-C]PYRIDINE AND PYRROLO[2,3-C]PYRIDINE DERIVATIVES AS SSAO INHIBITORS PNPO, SSB, XDH HCAR3 1797/4885HDAC3 1948/4885HDAC1 699/4885
US-10968223-B2 Imidazo[4,5-c]pyridine and pyrrolo[2,3-c]pyridine derivatives as SSAO inhibitors PNPO, PPOX, SCO2 HCAR3 2704/4885HDAC3 2167/4885HDAC1 1019/4885
US-20230110165-A1 Substituted Imidazo[4,5-c]pyridine Compounds and Compositions Thereof PNPO, XDH, EPX HCAR3 1754/4885HDAC3 629/4885HDAC1 481/4885
US-20200347059-A1 IMIDAZO[4,5-C]PYRIDINE AND PYRROLO[2,3-C]PYRIDINE DERIVATIVES AS SSAO INHIBITORS PNPO, PPOX, SCO2 HCAR3 2704/4885HDAC3 2167/4885HDAC1 1019/4885
US-20200262835-A1 COMPOUNDS QSOX1, AOX1, EPX HCAR3 1215/4885HDAC3 687/4885HDAC1 318/4885
US-20180194763-A1 IMIDAZO[4,5-C]PYRIDINE AND PYRROLO[2,3-C]PYRIDINE DERIVATIVES AS SSAO INHIBITORS PNPO, SSB, XDH HCAR3 1797/4885HDAC3 1948/4885HDAC1 699/4885
US-20150258101-A1 NEW COMPOUNDS AOX1, QSOX1, MAOB HCAR3 985/4885HDAC3 1827/4885HDAC1 562/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.