SCHEMBL16229778

SCHEMBL16229778

CN1C2C1C21Cc2cc(F)c(CCNS(=O)(=O)C3CCC3)cc2C1Cc1ccccc1

nearest known ligand 0.36

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
NR1D1 P20393 2/20 0.33
TBXAS1 P24557 1/20 0.33
HTR6 P50406 2/20 0.31
PKM P14618 1/20 0.31
SLC18A2 Q05940 1/20 0.30
ASAH1 Q13510 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16229754 0.93 RORC (0.32) NR1D1
SCHEMBL16784638 0.91 LMNA (0.34) NR1D1
SCHEMBL16229769 0.91 DPP4 (0.34) PKM
SCHEMBL16229795 0.90 GALR3 (0.35) NR1D1PKM
SCHEMBL16784635 0.87 SCN9A (0.35)
SCHEMBL16229782 0.86 SLC6A9 (0.39) HTR6PKM
SCHEMBL16229755 0.86 TBXAS1 (0.36) TBXAS1PKMSLC18A2
SCHEMBL16229759 0.84 RORC (0.33) HTR6
SCHEMBL16229784 0.83 DPP4 (0.34) PKM
SCHEMBL16229798 0.82 HTR6 (0.36) HTR6PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9051280-B2 Tetraline and indane derivatives, pharmaceutical compositions containing them, and their use in therapy AbbVie Deutschland GmbH & Co. KG (DE) 2015-06-09 US disclosed
US-8883839-B2 Tetraline and indane derivatives, pharmaceutical compositions containing them, and their use in therapy ABBOTT LABORATORIES (US) 2014-11-11 US disclosed