SCHEMBL1708201

SCHEMBL1708201

CC(=O)O[C@H]1c2ccc(NCc3cccc(-c4c(C)oc5cccnc45)c3C)cc2OC1C

nearest known ligand 0.33

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PDCD1 Q15116 1/20 0.33
CD274 Q9NZQ7 1/20 0.33
HDAC6 Q9UBN7 1/20 0.32
MAPT P10636 2/20 0.31
ALDH1A1 P00352 2/20 0.31
KDM4E B2RXH2 1/20 0.31
KMT2A Q03164 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
LMNA P02545 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1707845 0.88 PDCD1 (0.33) PDCD1CD274HDAC6MAPTALDH1A1
SCHEMBL3717530 0.85 FFAR1 (0.35) PDCD1CD274HDAC6MAPTALDH1A1
SCHEMBL13046194 0.79 FFAR1 (0.42) PDCD1CD274
SCHEMBL3721709 0.78 FFAR1 (0.46)
SCHEMBL1707908 0.78 CD274 (0.41) PDCD1CD274KMT2A
SCHEMBL1708437 0.78 PDCD1 (0.33) PDCD1CD274
SCHEMBL1707949 0.77 PDCD1 (0.36) PDCD1CD274MAPT
SCHEMBL1708101 0.77 RORC (0.33) PDCD1CD274
SCHEMBL1707867 0.75 ALDH1A1 (0.40) PDCD1CD274MAPTALDH1A1KDM4E
SCHEMBL10291390 0.75 FFAR1 (0.38) PDCD1CD274HDAC6MAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2440541-A1 NOVEL FUSED CYCLIC COMPOUND AND USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2012-04-18 EP disclosed