SCHEMBL1708225

SCHEMBL1708225

COc1ccc(-c2c(C)ccc(CNc3ccc4c(c3)OC(C)[C@H]4OC(C)=O)c2C)cn1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KLKB1 P03952 3/20 0.35
NTRK1 P04629 1/20 0.35
TNIK Q9UKE5 1/20 0.34
ALDH1A1 P00352 2/20 0.34
GAA P10253 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
FFAR1 O14842 1/20 0.33
RAB9A P51151 1/20 0.33
RECQL P46063 1/20 0.33
PIK3CA P42336 5/20 0.33
MTOR P42345 1/20 0.33
LMNA P02545 1/20 0.32
EZH2 Q15910 2/20 0.32
PDCD1 Q15116 1/20 0.32
CD274 Q9NZQ7 1/20 0.32
MAPT P10636 1/20 0.32
PIK3CD O00329 2/20 0.32
PIK3CB P42338 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1707908 0.89 CD274 (0.41) NTRK1TNIKRAB9APIK3CAEZH2
SCHEMBL1708467 0.85 FFAR1 (0.35) KLKB1NTRK1TNIKALDH1A1GAA
SCHEMBL1708599 0.84 WNT3A (0.38) RAB9AMTOREZH2MAPT
SCHEMBL1708592 0.82 ALDH1A1 (0.33) ALDH1A1GAASMN1; SMN2TDP1L3MBTL1
SCHEMBL1707989 0.81 EED (0.38) ALDH1A1GAASMN1; SMN2MTOREZH2
SCHEMBL1708222 0.80 STAT6 (0.36) GAAMTOREZH2
SCHEMBL1708466 0.78 FFAR1 (0.49) FFAR1
SCHEMBL1708221 0.77 INSR (0.34) ALDH1A1GAASMN1; SMN2TDP1L3MBTL1
SCHEMBL1708277 0.77 RORC (0.33)
SCHEMBL1707867 0.76 ALDH1A1 (0.40) ALDH1A1GAASMN1; SMN2TDP1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2440541-A1 NOVEL FUSED CYCLIC COMPOUND AND USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2012-04-18 EP disclosed
WO-2010143733-A1 NOVEL FUSED CYCLIC COMPOUND AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-12-16 WO disclosed