SCHEMBL1748249

SCHEMBL1748249

Fc1cc(F)c2nc(Cl)sc2c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 9/20 0.56
MAPT P10636 8/20 0.56
MEN1 O00255 6/20 0.56
KMT2A Q03164 6/20 0.56
ALDH1A1 P00352 5/20 0.56
PKM P14618 3/20 0.56
TDP1 Q9NUW8 3/20 0.56
SMN1; SMN2 Q16637 5/20 0.51
NPC1 O15118 9/20 0.50
HPGD P15428 1/20 0.49
HTT P42858 3/20 0.47
KDM4E B2RXH2 2/20 0.47
MCL1 Q07820 2/20 0.47
NPSR1 Q6W5P4 1/20 0.47
POLB P06746 1/20 0.44
THRB P10828 1/20 0.44
RECQL P46063 1/20 0.44
BLM P54132 1/20 0.44
LMNA P02545 3/20 0.43
AGTR1 P30556 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8331402 0.84 ALDH1A1 (0.43) RAB9AMAPTMEN1KMT2AALDH1A1
SCHEMBL23290946 0.84 ALDH1A1 (0.43) RAB9AMAPTMEN1KMT2AALDH1A1
SCHEMBL12210694 0.81 NSD1 (0.39) RAB9AMAPTMEN1KMT2AALDH1A1
SCHEMBL19783572 0.78 RAB9A (0.62) RAB9AMAPTMEN1KMT2AALDH1A1
SCHEMBL2615996 0.76 RAB9A (0.56) RAB9AMAPTMEN1KMT2AALDH1A1
SCHEMBL474219 0.76 ALDH1A1 (0.61) RAB9AMAPTMEN1KMT2AALDH1A1
SCHEMBL335937 0.76 ALDH1A1 (0.61) RAB9AMAPTMEN1KMT2AALDH1A1
SCHEMBL20554157 0.75 NR1H4 (0.39) LMNAGAA
SCHEMBL2634141 0.72 SMN1; SMN2 (0.61) RAB9AMAPTMEN1KMT2AALDH1A1
SCHEMBL13439534 0.72 RAB9A (0.51) RAB9AMAPTMEN1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 64 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117120423-B Indolylamine 2, 3-dioxygenase inhibitors, methods of preparing the same, and pharmaceutical compositions containing the same 柳韩洋行 2026-02-27 CN disclosed
EP-4015510-B1 ANTI-TUMOUR COMPOUND BASED ON JWA GENE ACTIVATION AND HER2 DEGRADATION, PREPARATION METHOD THEREFOR, AND USE THEREOF Simcere pharmaceutical co ltd (CN) 2025-08-20 EP disclosed
US-20250011293-A1 LEUKOTRIENE SYNTHESIS INHIBITORS NAEGIS PHARMACEUTICALS INC. (CA) 2025-01-09 US disclosed
US-20240174636-A1 NOVEL INDOLEAMINE 2,3-DIOXYGENASE INHIBITORS, PROCESSES FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITIONS COMPRISING THE SAME YUHAN CORPORATION (KR) 2024-05-30 US disclosed
US-11976052-B2 Leukotriene synthesis inhibitors NAEGIS PHARMACEUTICALS INC. (CA) 2024-05-07 US disclosed
EP-4313965-A1 NOVEL INDOLEAMINE 2,3-DIOXYGENASE INHIBITORS, PROCESSES FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITIONS COMPRISING THE SAME Yuhan Corporation (KR) 2024-02-07 EP disclosed
CN-117120423-A Novel indoleamine 2,3-dioxygenase inhibitors, process for preparing the same and pharmaceutical compositions containing the same 柳韩洋行 2023-11-24 CN disclosed
WO-2022203332-A1 NOVEL INDOLEAMINE 2,3-DIOXYGENASE INHIBITORS, PROCESSES FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITIONS COMPRISING THE SAME YUHAN CORPORATION (KR) 2022-09-29 WO disclosed
US-11427575-B2 Antitumor compound for activating JWA gene and degrading HER2, preparation method thereof, and application thereof SIMCERE PHARMACEUTICAL CO., LTD. (CN) 2022-08-30 US disclosed
EP-4015510-A1 ANTI-TUMOUR COMPOUND BASED ON JWA GENE ACTIVATION AND HER2 DEGRADATION, PREPARATION METHOD THEREFOR, AND USE THEREOF Simcere Pharmaceutical Co. Ltd. (CN) 2022-06-22 EP disclosed
WO-2004100881-A2 PREPARATION AND USE OF ARYL ALKYL ACID DERIVATIVES FOR THE TREATMENT OF OBESITY BAYER PHARMACEUTICALS CORPORATION (US) 2004-11-25 WO disclosed
US-20040224997-A1 Preparation and use of aryl alkyl acid derivatives for the treatment of obesity BAYER PHARMACEUTICALS CORPORATION 2004-11-11 US disclosed
EP-1087962-A4 PREPARATION OF HETEROARYL COMPOUNDS LILLY CO ELI (US) 2001-10-04 EP disclosed
EP-1087962-A1 PREPARATION OF HETEROARYL COMPOUNDS ELI LILLY AND COMPANY (US) 2001-04-04 EP disclosed
WO-1999065896-A1 PREPARATION OF HETEROARYL COMPOUNDS ELI LILLY AND COMPANY (US) 1999-12-23 WO disclosed
EP-0060426-B1 N-(2,2,2-TRIFLUOROETHYL)-N-ALKYL-AZOLYLOXYACETIC-ACID AMIDES, THEIR PREPARATION AND USE AS HERBICIDES AND INTERMEDIATES FOR THEIR PREPARATION BAYER AG (DE) 1986-04-23 EP disclosed
US-4465504-A Herbicidally active novel N-(2,2,2-trifluoroethyl)-N-alkyl-azolyloxyacetic acid amides and intermediates therefor BAYER AKTIENGESELLSCHAFT (DE) 1984-08-14 US disclosed
US-4455428-A HERBICIDES BAYER AKTIENGESELLSCHAFT (DE) 1984-06-19 US disclosed
US-4408055-A HERBICIDES BAYER AKTIENGESELLSCHAFT (DE) 1983-10-04 US disclosed
EP-0081730-A1 Process for the preparation of hetaryloxyacetamides BAYER AG (DE) 1983-06-22 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240174636-A1 NOVEL INDOLEAMINE 2,3-DIOXYGENASE INHIBITORS, PROCESSES FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITIONS COMPRISING THE SAME IDO1, IDO2, INMT RAB9A 2470/4885MAPT 2422/4885MEN1 3028/4885
US-20040224997-A1 Preparation and use of aryl alkyl acid derivatives for the treatment of obesity FABP4, GPR119, LIPC RAB9A 2066/4885MAPT 4379/4885MEN1 4348/4885
US-11427575-B2 Antitumor compound for activating JWA gene and degrading HER2, preparation method thereof, and application thereof EGFR, ERBB2, ERBB3 RAB9A 1648/4885MAPT 4856/4885MEN1 2781/4885
US-11976052-B2 Leukotriene synthesis inhibitors LTC4S, LTB4R2, LTA4H RAB9A 4666/4885MAPT 3739/4885MEN1 3388/4885
US-20250011293-A1 LEUKOTRIENE SYNTHESIS INHIBITORS LTC4S, LTB4R2, LTA4H RAB9A 4666/4885MAPT 3739/4885MEN1 3388/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.