SCHEMBL181807

SCHEMBL181807

CC(C)(C)OC(=O)N[C@H](CCc1ccccc1)C(=O)O

nearest known ligand 0.71

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CTSK P43235 5/20 0.71
CTSS P25774 5/20 0.71
PPARA Q07869 5/20 0.62
PPARG P37231 4/20 0.62
ACE P12821 1/20 0.60
CTSB P07858 2/20 0.56
CTSL P07711 1/20 0.56
PPARD Q03181 2/20 0.56
ATM Q13315 1/20 0.52
IDO1 P14902 1/20 0.51
APP P05067 1/20 0.51
SCN9A Q15858 1/20 0.51
ALDH1A1 P00352 1/20 0.50
TSHR P16473 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL181775 1.00 CTSK (0.71) CTSKCTSSPPARAPPARGACE
SCHEMBL181808 1.00 CTSK (0.71) CTSKCTSSPPARAPPARGACE
SCHEMBL8238590 0.95 PPARA (0.70) CTSKCTSSPPARAPPARGACE
SCHEMBL13744253 0.95 PPARA (0.70) CTSKCTSSPPARAPPARGACE
SCHEMBL344068 0.93 CTSK (0.63) CTSKCTSSPPARAPPARGACE
SCHEMBL22651626 0.93 CTSK (0.63) CTSKCTSSPPARAPPARGACE
SCHEMBL19605638 0.93 CTSK (0.63) CTSKCTSSPPARAPPARGACE
SCHEMBL2781406 0.92 CTSK (0.63) CTSKCTSSPPARAPPARGACE
SCHEMBL1374859 0.92 CTSK (0.63) CTSKCTSSPPARAPPARGACE
SCHEMBL346311 0.92 CTSK (0.63) CTSKCTSSPPARAPPARGACE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 292 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260125390-A1 SOLID FORMS OF MACROCYCLIC COMPOUNDS, SALTS AND FORMULATIONS THEREOF, AND METHODS OF PREPARING AND USING THE SAME KURA ONCOLOGY INC (US) 2026-05-07 US disclosed
EP-4720073-A1 SOLID FORMS OF A MACROCYCLIC FARNESYLTRANSFERASE INHIBITOR AND FORMULATIONS THEREOF, AND METHODS OF PREPARING AND USING THE MACROCYCLIC COMPOUND AND ITS SOLID FORMS Kura Oncology, Inc. (US) 2026-04-08 EP disclosed
EP-3788039-B1 FACTOR XIIA INHIBITORS UNIV LEEDS INNOVATIONS LTD (GB) 2026-02-11 EP disclosed
US-20260001924-A1 NEMO COILED COIL MIMICS AND METHODS OF USING SAME NEW YORK UNIVERSITY (US) 2026-01-01 US disclosed
US-20250376443-A1 MASP-2 INHIBITORS AND METHODS OF USE OMEROS CORPORATION (US) 2025-12-11 US disclosed
US-20250368604-A1 MASP-2 INHIBITORS AND METHODS OF USE OMEROS CORPORATION (US) 2025-12-04 US disclosed
US-12466835-B1 Solid forms of macrocyclic compounds, salts and formulations thereof, and methods of preparing and using the same KURA ONCOLOGY, INC. (US) 2025-11-11 US disclosed
US-12384757-B2 Methods of synthesizing substituted pyridinone-pyridinyl compounds ACLARIS THERAPEUTICS, INC. (US) 2025-08-12 US disclosed
US-12371461-B2 Nemo coiled coil mimics and methods of using same NEW YORK UNIVERSITY (US) 2025-07-29 US disclosed
US-12336991-B2 Factor XIIA inhibitors UNIVERSITY OF LEEDS (GB) 2025-06-24 US disclosed
US-5206235-A Animal growth regulators; stimulants MERCK & CO., INC. (US) 1993-04-27 US disclosed
EP-0480969-A4 AMINO ACID ANALOG CCK ANTAGONISTS 1993-01-07 EP disclosed
EP-0513974-A1 Novel benzo-fused lactams that promote the release of growth hormone MERCK & CO. INC. (US) 1992-11-19 EP disclosed
WO-1992016524-A1 BENZO-FUSED LACTAMS PROMOTE RELEASE OF GROWTH HORMONE MERCK & CO., INC. (US) 1992-10-01 WO disclosed
US-5149795-A Fungicides BAYER AG (DE) 1992-09-22 US disclosed
EP-0480969-A1 AMINO ACID ANALOG CCK ANTAGONISTS ABBOTT LABORATORIES (US) 1992-04-22 EP disclosed
EP-0478362-A2 Fibrinogen receptor antagonists MERCK & CO. INC. (US) 1992-04-01 EP disclosed
US-5019560-A Method for treating fungal infections with nikkomycin derivatives BAYER AG (DE) 1991-05-28 US disclosed
WO-1991000725-A2 AMINO ACID ANALOG CCK ANTAGONISTS ABBOTT LABORATORIES (US) 1991-01-24 WO disclosed
EP-0367954-A1 Nikkomycin derivatives, antimycotic compositions of nikkomycin derivatives and azole antimycotics BAYER AG (DE) 1990-05-16 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20260125390-A1 SOLID FORMS OF MACROCYCLIC COMPOUNDS, SALTS AND FORMULATIONS THEREOF, AND METHODS OF PREPARING AND USING THE SAME FDPS, PCTP, MTTP CTSK 2131/4885CTSS 517/4885PPARA 740/4885
US-12466835-B1 Solid forms of macrocyclic compounds, salts and formulations thereof, and methods of preparing and using the same FNTA, SF3B1, SF3A1 CTSK 3833/4885CTSS 3207/4885PPARA 1562/4885
US-12384757-B2 Methods of synthesizing substituted pyridinone-pyridinyl compounds PIR, PUM1, ZRANB2 CTSK 3919/4885CTSS 3313/4885PPARA 1389/4885
US-12371461-B2 Nemo coiled coil mimics and methods of using same COIL, CALCOCO2, NCAPH CTSK 4487/4885CTSS 4120/4885PPARA 4497/4885
US-20250368604-A1 MASP-2 INHIBITORS AND METHODS OF USE MASP2, METAP2, SPINT2 CTSK 485/4885CTSS 439/4885PPARA 4706/4885
US-20250376443-A1 MASP-2 INHIBITORS AND METHODS OF USE MASP2, METAP2, SPINT2 CTSK 436/4885CTSS 379/4885PPARA 4696/4885
US-20260001924-A1 NEMO COILED COIL MIMICS AND METHODS OF USING SAME DDX21, PHAX, RBX1 CTSK 4676/4885CTSS 4503/4885PPARA 3778/4885
US-12336991-B2 Factor XIIA inhibitors F11, F13B, F12 CTSK 303/4885CTSS 714/4885PPARA 4768/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.